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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Fibroblast growth factor receptor 3 | ||
| Ligand | BDBM130067 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | LanthaScreen TR-FRET Assay | ||
| Temperature | 298.15±n/a K | ||
| IC50 | >10000±n/a nM | ||
| Comments | extracted | ||
| Citation |  Furet, P; Graus Porta, D; Guagnano, V Quinoline carboxamide derivatives as protein tyrosine kinase inhibitors US Patent US8815901 Publication Date 8/26/2014 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Fibroblast growth factor receptor 3 | |||
| Name: | Fibroblast growth factor receptor 3 | ||
| Synonyms: | CD_antigen: CD333 | FGFR-3 | FGFR3 | FGFR3_HUMAN | Fibroblast growth factor receptor | Fibroblast growth factor receptor 3 (FGFR3) | JTK4 | ||
| Type: | Protein | ||
| Mol. Mass.: | 87699.57 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | P22607 | ||
| Residue: | 806 | ||
| Sequence: |
| ||
| BDBM130067 | |||
| n/a | |||
| Name | BDBM130067 | ||
| Synonyms: | US8815901, 17 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C19H14Cl2N6O3 | ||
| Mol. Mass. | 445.259 | ||
| SMILES | COc1cc(OC)c(Cl)c(c1Cl)-c1ccc(C(=O)Nc2ncn[nH]2)c2nccnc12 |(5.31,3.91,;6.08,2.57,;5.31,1.24,;6.08,-.1,;5.31,-1.43,;6.08,-2.76,;7.62,-2.76,;3.77,-1.43,;3,-2.76,;3,-.1,;3.77,1.24,;3,2.57,;1.46,-.1,;.69,1.24,;-.85,1.24,;-1.62,-.1,;-3.16,-.1,;-3.93,1.24,;-3.93,-1.43,;-5.47,-1.43,;-6.38,-.18,;-7.84,-.66,;-7.84,-2.2,;-6.38,-2.67,;-.85,-1.43,;-1.62,-2.76,;-.85,-4.1,;.69,-4.1,;1.46,-2.76,;.69,-1.43,)| | ||
| Structure | 
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