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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Neuropeptide Y receptor type 5 | ||
| Ligand | BDBM141361 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Binding Assay | ||
| pH | 7.4±n/a | ||
| Temperature | 298.15±n/a K | ||
| IC50 | 0.61±n/a nM | ||
| Citation |  Hayashi, K; Tamura, Y; Omori, N 5-membered ring heteroaromatic derivatives having NPY Y5 receptor antagonistic activity US Patent US8916594 Publication Date 12/23/2014 | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| Neuropeptide Y receptor type 5 | |||
| Name: | Neuropeptide Y receptor type 5 | ||
| Synonyms: | NPY-Y5 | NPY5R_MOUSE | Neuropeptide Y receptor Y5 | Neuropeptide Y receptor type 5 (NPY Y5) | Npy5 | Npy5r | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 52807.91 | ||
| Organism: | Mus musculus (Mouse) | ||
| Description: | O70342 | ||
| Residue: | 466 | ||
| Sequence: |
| ||
| BDBM141361 | |||
| n/a | |||
| Name | BDBM141361 | ||
| Synonyms: | US8916594, I-147 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C17H28F2N4O3S | ||
| Mol. Mass. | 406.491 | ||
| SMILES | CC(C)S(=O)(=O)NC[C@H]1CC[C@@H](CC1)Nc1nc(no1)C1(C)CC(F)(F)C1 |r,wU:8.7,wD:11.14,(-9.71,.87,;-8.38,.1,;-8.38,-1.44,;-7.04,.87,;-7.81,2.21,;-6.27,2.21,;-5.71,.1,;-4.38,.87,;-3.04,.1,;-1.71,.87,;-.38,.1,;-.38,-1.44,;-1.71,-2.21,;-3.04,-1.44,;.96,-2.21,;2.29,-1.44,;3.76,-1.91,;4.66,-.67,;3.76,.58,;2.29,.1,;6.2,-.67,;5.43,.67,;7.29,-1.76,;8.38,-.67,;9.71,.1,;9.71,-1.44,;7.29,.42,)| | ||
| Structure | 
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