| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 3 |
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| Ligand | BDBM223533 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Calcium Flux Assay Using Fluorometric Imaging Plate Reader (FLIPR) Assay |
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| Temperature | 298.15±n/a K |
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| IC50 | >30000±n/a nM |
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| Comments | extracted |
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| Citation |  Gabriel, SD; Hamilton, MM; Lucas, MC; Qian, Y; Sidduri, A N-alkyltriazole compounds as LPAR antagonists US Patent US9321738 Publication Date 4/26/2016 |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 3 |
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| Name: | Lysophosphatidic acid receptor 3 |
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| Synonyms: | EDG7 | LPA3 | LPAR3 | LPAR3_HUMAN | Lysophosphatidic acid receptor 1/3 | Lysophosphatidic acid receptor 3 (LPAR3) | Lysophosphatidic acid receptor Edg-7 |
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| Type: | Enzyme |
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| Mol. Mass.: | 40149.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9UBY5 |
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| Residue: | 353 |
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| Sequence: | MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
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| BDBM223533 |
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| n/a |
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| Name | BDBM223533 |
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| Synonyms: | US9321738, 10 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H27FN4O4 |
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| Mol. Mass. | 514.5475 |
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| SMILES | COC(=O)C1(CC1)c1ccc(cc1)-c1ccc(-c2nnn(C)c2NC(=O)O[C@H](C)c2ccccc2)c(F)c1 |r| |
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| Structure | 
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