| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Peroxisome proliferator-activated receptor delta |
|---|
| Ligand | BDBM232296 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Kinase Activity Assay |
|---|
| EC50 | 331±n/a nM |
|---|
| Citation |  Wang, Y; Zheng, G; Sun, P; Li, Y; Wu, Y; Liu, B; Liu, X; Bai, H; Li, H; Zheng, X Compounds having activating effect on subtypes of peroxisome proliferator-activated receptors and its preparation method and uses US Patent US9346770 Publication Date 5/24/2016 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Peroxisome proliferator-activated receptor delta |
|---|
| Name: | Peroxisome proliferator-activated receptor delta |
|---|
| Synonyms: | NR1C2 | NUC1 | NUCI | Nuclear hormone receptor 1 | Nuclear receptor subfamily 1 group C member 2 | PPAR delta | PPAR-beta | PPARB | PPARD | PPARD_HUMAN | Peroxisome proliferator-activated receptor | Peroxisome proliferator-activated receptor beta | Peroxisome proliferator-activated receptor delta |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 49910.45 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q03181 |
|---|
| Residue: | 441 |
|---|
| Sequence: | MEQPQEEAPEVREEEEKEEVAEAEGAPELNGGPQHALPSSSYTDLSRSSSPPSLLDQLQM
GCDGASCGSLNMECRVCGDKASGFHYGVHACEGCKGFFRRTIRMKLEYEKCERSCKIQKK
NRNKCQYCRFQKCLALGMSHNAIRFGRMPEAEKRKLVAGLTANEGSQYNPQVADLKAFSK
HIYNAYLKNFNMTKKKARSILTGKASHTAPFVIHDIETLWQAEKGLVWKQLVNGLPPYKE
ISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNK
DGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGD
RPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRI
KKTETETSLHPLLQEIYKDMY
|
|
|
|---|
| BDBM232296 |
|---|
| n/a |
|---|
| Name | BDBM232296 |
|---|
| Synonyms: | US9346770, 9 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H25N3O5 |
|---|
| Mol. Mass. | 423.4617 |
|---|
| SMILES | CCc1cc(OCCc2nc(oc2C)-c2ccc(cc2)C(N)=O)ncc1CCC(O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
