| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
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| Ligand | BDBM234291 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | CB1 Receptor Binding Assay (In Vitro) |
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| IC50 | >1000±n/a nM |
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| Citation |  Tu, G; Xiong, F; Huang, H; Kuang, B; Li, S Design, synthesis and biological evaluation of CB1 cannabinoid receptor ligands derived from the 1,5-diarylpyrazole scaffold. J Enzyme Inhib Med Chem26:222-30 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 1 |
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| Name: | Cannabinoid receptor 1 |
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| Synonyms: | CNR1 | Cannabinoid receptor 1 (CB1) |
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| Type: | Protein |
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| Mol. Mass.: | 37458.12 |
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| Organism: | Cricetulus griseus (Chinese hamster) |
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| Description: | Q99NU1 |
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| Residue: | 331 |
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| Sequence: | FRGSPFQEKMTAGDNSQLVPVVDTTNITEFYNKSLSSYKENEENIQCGENFMDMECFMIL
NPSQQLAIAVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFV
YSFVDFHVFHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRP
KAVVAFCLMWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIV
YAYMYILWKAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVV
LIICWGPLLAIMVYDVFGKMNKLIKTVFAFC
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| BDBM234291 |
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| n/a |
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| Name | BDBM234291 |
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| Synonyms: | [2-[(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazol-3-yl]methoxy]propionic acid (14d) |
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| Type | Small organic molecule |
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| Emp. Form. | C19H15Cl3N2O3 |
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| Mol. Mass. | 425.693 |
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| SMILES | CC(Oc1nn(c(c1C)-c1ccc(Cl)cc1)-c1ccc(Cl)cc1Cl)C(O)=O |
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| Structure | 
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