| Reaction Details |
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 | Report a problem with these data |
| Target | Mast/stem cell growth factor receptor Kit [544-976] |
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| Ligand | BDBM239033 |
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| Substrate/Competitor | BioDB n*138 SEQ ID NO: 2 |
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| Meas. Tech. | Biochemical Assay |
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| pH | 7.9±n/a |
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| IC50 | 61±n/a nM |
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| Comments | extracted |
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| Citation |  Lombardi Borgia, A; Ciomei, M; Donati, D; Nesi, M Substituted indazole derivatives active as kinase inhibitors US Patent US9408850 Publication Date 8/9/2016 |
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| More Info.: | Get all data from this article, Assay Method |
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| Mast/stem cell growth factor receptor Kit [544-976] |
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| Name: | Mast/stem cell growth factor receptor Kit [544-976] |
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| Synonyms: | KIT | KIT_HUMAN | SCFR | Tyrosine-protein kinase Kit |
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| Type: | Protein |
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| Mol. Mass.: | 48998.23 |
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| Organism: | Homo sapiens (Human) |
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| Description: | aa 544-976 |
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| Residue: | 433 |
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| Sequence: | TYKYLQKPMYEVQWKVVEEINGNNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKV
VEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIG
GPTLVITEYCCYGDLLNFLRRKRDSFICSKQEDHAEAALYKNLLHSKESSCSDSTNEYMD
MKPGVSYVVPTKADKRRSVRIGSYIERDVTPAIMEDDELALDLEDLLSFSYQVAKGMAFL
ASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVVKGNARLPVKWMAPESIFN
CVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIM
KTCWDADPLKRPTFKQIVQLIEKQISESTNHIYSNLANCSPNRQKPVVDHSVRINSVGST
ASSSQPLLVHDDV
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| BDBM239033 |
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| BioDB n*138 SEQ ID NO: 2 |
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| Name: | BioDB n*138 SEQ ID NO: 2 |
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| Synonyms: | n/a |
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| Type: | Peptide Substrate |
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| Mol. Mass.: | 3822.64 |
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| Organism: | Artificial Organism |
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| Description: | SEQ ID NO: 2 |
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| Residue: | 30 |
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| Sequence: | KWEEINGNNYVYIDPTQLPYDHKWEFPRNR
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