| Reaction Details |
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 | Report a problem with these data |
| Target | Urokinase-type plasminogen activator |
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| Ligand | BDBM240796 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Urokinase Amidolytic Assay |
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| pH | 8.8±n/a |
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| Ki | 275600±21900 nM |
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| Comments | extracted |
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| Citation |  Markowska, A; Bruzgo, M; Surazynski, A; Midura-Nowaczek, K Tripeptides with non-code amino acids as potential serine proteases inhibitors. J Enzyme Inhib Med Chem28:639-43 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Urokinase-type plasminogen activator |
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| Name: | Urokinase-type plasminogen activator |
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| Synonyms: | 3.4.21.73 | PLAU | U-plasminogen activator | UROK_HUMAN | Urokinase | Urokinase-type plasminogen activator (uPA) | Urokinase-type plasminogen activator chain B | Urokinase-type plasminogen activator long chain A | Urokinase-type plasminogen activator short chain A | Urokinase-type plasminogen activator/surface receptor | uPA |
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| Type: | Enzyme |
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| Mol. Mass.: | 48528.62 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P00749 |
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| Residue: | 431 |
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| Sequence: | MRALLARLLLCVLVVSDSKGSNELHQVPSNCDCLNGGTCVSNKYFSNIHWCNCPKKFGGQ
HCEIDKSKTCYEGNGHFYRGKASTDTMGRPCLPWNSATVLQQTYHAHRSDALQLGLGKHN
YCRNPDNRRRPWCYVQVGLKLLVQECMVHDCADGKKPSSPPEELKFQCGQKTLRPRFKII
GGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLG
RSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICL
PSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKML
CAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIR
SHTKEENGLAL
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| BDBM240796 |
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| n/a |
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| Name | BDBM240796 |
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| Synonyms: | H-D-Ser-αMePhe-Arg-OH (7) |
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| Type | Small organic molecule |
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| Emp. Form. | C20H32N6O4 |
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| Mol. Mass. | 420.5059 |
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| SMILES | CC[C@@H](N)C(=O)N[C@@](C)(Cc1ccccc1)C(=O)N[C@H](CCCNC(N)=N)C(O)=O |r| |
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| Structure | 
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