| Reaction Details |
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 | Report a problem with these data |
| Target | Ryanodine receptor 1 [4317-4329] |
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| Ligand | BDBM430064 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | QSS Assist FP assay |
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| IC50 | 1.80±n/a nM |
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| Citation |  Sugimoto, T; Sakamoto, T; Yamamoto, F; Kobayakawa, Y; Egashira, N; Ichikawa, K; Machida, T 5H-pyrrolo[2,3-D]pyrimidin-6(7H)-one derivative US Patent US10538528 Publication Date 1/21/2020 |
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| More Info.: | Get all data from this article, Assay Method |
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| Ryanodine receptor 1 [4317-4329] |
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| Name: | Ryanodine receptor 1 [4317-4329] |
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| Synonyms: | Biotinylated Substrate Peptide | RYDR | RYR1 | RYR1_HUMAN |
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| Type: | Peptide |
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| Mol. Mass.: | 2871.44 |
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| Organism: | n/a |
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| Description: | P21817[4317-4329] |
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| Residue: | 24 |
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| Sequence: | biotin-C6linker-VRRLRRLTAREAA
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| BDBM430064 |
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| n/a |
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| Name | BDBM430064 |
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| Synonyms: | US10538528, Compound 12 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H33FN8O |
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| Mol. Mass. | 504.6023 |
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| SMILES | CCNCCNc1ccc(nc1C1CCN(CC1)c1ncnc2NC(=O)C(C)(C)c12)-c1cncc(F)c1 |
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| Structure | 
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