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TargetRetinaldehyde-binding protein 1
LigandBDBM323419
Substrate/Competitorn/a
Meas. Tech.In Vitro Isomerase Inhibition Assay
IC50<100.0±n/a nM
Citation Scott, ILKuksa, VAOrme, MWLittle, Jr., TLGall, AHong, F Alkoxy compounds for disease treatment US Patent US10639286 Publication Date 5/5/2020
More Info.:Get all data from this article,  Assay Method
 
Retinaldehyde-binding protein 1
Name:Retinaldehyde-binding protein 1
Synonyms:CRALBP | Cellular retinaldehyde-binding protein | RLBP1 | RLBP1_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:36462.25
Organism:Homo sapiens (Human)
Description:P12271
Residue:317
Sequence:
MSEGVGTFRMVPEEEQELRAQLEQLTTKDHGPVFGPCSQLPRHTLQKAKDELNEREETRE
EAVRELQEMVQAQAASGEELAVAVAERVQEKDSGFFLRFIRARKFNVGRAYELLRGYVNF
RLQYPELFDSLSPEAVRCTIEAGYPGVLSSRDKYGRVVMLFNIENWQSQEITFDEILQAY
CFILEKLLENEETQINGFCIIENFKGFTMQQAASLRTSDLRKMVDMLQDSFPARFKAIHF
IHQPWYFTTTYNVVKPFLKSKLLERVFVHGDDLSGFYQEIDENILPSDFGGTLPKYDGKA
VAEQLFGPQAQAENTAF
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM323419
n/a
NameBDBM323419
Synonyms:(R)-3-Amino-1-(3-(Cyclohexylmethoxy)Phenyl)Propan-1-Ol | US10188615, Example 28 | US10639286, Example 28
TypeSmall organic molecule
Emp. Form.C16H25NO2
Mol. Mass.263.3752
SMILESNCC[C@@H](O)c1cccc(OCC2CCCCC2)c1 |r|
Structure
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