| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 3 |
|---|
| Ligand | BDBM311875 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Radioligand Binding Assays |
|---|
| Ki | >8580±n/a nM |
|---|
| Citation |  Giovannini, R; Cui, Y; Doods, H; Ferrara, M; Just, S; Kuelzer, R; Lingard, I; Mazzaferro, R; Rudolf, K Somatostatin receptor subtype 4 (SSTR4) agonists US Patent US10675268 Publication Date 6/9/2020 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 3 |
|---|
| Name: | Somatostatin receptor type 3 |
|---|
| Synonyms: | SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3) |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 45855.97 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P32745 |
|---|
| Residue: | 418 |
|---|
| Sequence: | MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLL
GNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVM
AVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVV
FSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRV
WAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVA
LPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEE
SREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
|
|
|
|---|
| BDBM311875 |
|---|
| n/a |
|---|
| Name | BDBM311875 |
|---|
| Synonyms: | US10166214, Example 11 | US10675268, Example 11 | US9789082, Example 11 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H19ClN4O |
|---|
| Mol. Mass. | 318.801 |
|---|
| SMILES | CC(C)(NC(=O)[C@@H]1[C@H]2CNC[C@@H]12)c1nc2ccc(Cl)cc2[nH]1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
