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TargetOxidized low-density lipoprotein receptor 1
LigandBDBM50232678
Substrate/Competitorn/a
Meas. Tech.Inhibition Assay
IC50>1000000±n/a nM
Citation Findlay, ADTurner, CIDeodhar, MFoot, JSJarolimek, WZhou, WRobertson, AD Indole and azaindole haloallylamine derivative inhibitors of lysyl oxidases and uses thereof US Patent US10717734 Publication Date 7/21/2020
More Info.:Get all data from this article,  Assay Method
 
Oxidized low-density lipoprotein receptor 1
Name:Oxidized low-density lipoprotein receptor 1
Synonyms:LOX-1 | LOX1 | Lectin-like oxLDL receptor 1 | Lectin-like oxidized LDL receptor 1 | Lectin-type oxidized LDL receptor 1 | OLR1 | OLR1_BOVIN | Ox-LDL receptor 1 | bLOX-1
Type:Protein
Mol. Mass.:30894.65
Organism:Bovine
Description:P79391
Residue:270
Sequence:
MTVDDPKGMKDQLDQKPNGKTAKGFVSSWRWYPAAVTLGVLCLGLLVTVILLILQLSQVS
DLIKKQQANITHQEDILEGQILAQRRSEKSAQESQKELKEMIETLAHKLDEKSKKLMELH
RQNLNLQEVLKEAANYSGPCPQDWLWHEENCYQFSSGSFNWEKSQENCLSLDAHLLKINS
TDELEFIQQMIAHSSFPFWMGLSMRKPNYSWLWEDGTPLTPHLFRIQGAVSRMYPSGTCA
YIQRGTVFAENCILTAFSICQKKANLLRAQ
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  Blast E-value cutoff:
BDBM50232678
n/a
NameBDBM50232678
Synonyms:CHEBI:27413 | CHEMBL1618272 | US10717734, Compound BAPN | US11098045, Compound BAPN
TypeSmall organic molecule
Emp. Form.C3H6N2
Mol. Mass.70.0931
SMILESNCCC#N
Structure
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