| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Oxidized low-density lipoprotein receptor 1 |
|---|
| Ligand | BDBM454336 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Inhibition Assay |
|---|
| IC50 | >300000±n/a nM |
|---|
| Citation |  Findlay, AD; Turner, CI; Deodhar, M; Foot, JS; Jarolimek, W; Zhou, W; Robertson, AD Indole and azaindole haloallylamine derivative inhibitors of lysyl oxidases and uses thereof US Patent US10717734 Publication Date 7/21/2020 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Oxidized low-density lipoprotein receptor 1 |
|---|
| Name: | Oxidized low-density lipoprotein receptor 1 |
|---|
| Synonyms: | LOX-1 | LOX1 | Lectin-like oxLDL receptor 1 | Lectin-like oxidized LDL receptor 1 | Lectin-type oxidized LDL receptor 1 | OLR1 | OLR1_BOVIN | Ox-LDL receptor 1 | bLOX-1 |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 30894.65 |
|---|
| Organism: | Bovine |
|---|
| Description: | P79391 |
|---|
| Residue: | 270 |
|---|
| Sequence: | MTVDDPKGMKDQLDQKPNGKTAKGFVSSWRWYPAAVTLGVLCLGLLVTVILLILQLSQVS
DLIKKQQANITHQEDILEGQILAQRRSEKSAQESQKELKEMIETLAHKLDEKSKKLMELH
RQNLNLQEVLKEAANYSGPCPQDWLWHEENCYQFSSGSFNWEKSQENCLSLDAHLLKINS
TDELEFIQQMIAHSSFPFWMGLSMRKPNYSWLWEDGTPLTPHLFRIQGAVSRMYPSGTCA
YIQRGTVFAENCILTAFSICQKKANLLRAQ
|
|
|
|---|
| BDBM454336 |
|---|
| n/a |
|---|
| Name | BDBM454336 |
|---|
| Synonyms: | US10717734, Compound 12 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H24FN3O2S |
|---|
| Mol. Mass. | 401.498 |
|---|
| SMILES | Cc1c(Cc2ccc(cc2)S(C)(=O)=O)c2nc(C)ccc2n1C\C(F)=C\CN |
|---|
| Structure | 
|
|---|
Search and Browse
