| Reaction Details |
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 | Report a problem with these data |
| Target | Free fatty acid receptor 1 |
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| Ligand | BDBM301754 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Pharmacological Assay |
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| EC50 | 7.00±n/a nM |
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| Citation |  Eckhardt, M; Frattini, S; Langkopf, E; Wagner, H Indanyloxydihydrobenzofuranylacetic acids US Patent US9597310 Publication Date 3/21/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Free fatty acid receptor 1 |
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| Name: | Free fatty acid receptor 1 |
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| Synonyms: | FFAR1 | FFAR1_HUMAN | G-protein Coupled Receptor 40 | GPR40 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 31473.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | O14842 |
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| Residue: | 300 |
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| Sequence: | MDLPPQLSFGLYVAAFALGFPLNVLAIRGATAHARLRLTPSLVYALNLGCSDLLLTVSLP
LKAVEALASGAWPLPASLCPVFAVAHFFPLYAGGGFLAALSAGRYLGAAFPLGYQAFRRP
CYSWGVCAAIWALVLCHLGLVFGLEAPGGWLDHSNTSLGINTPVNGSPVCLEAWDPASAG
PARFSLSLLLFFLPLAITAFCYVGCLRALARSGLTHRRKLRAAWVAGGALLTLLLCVGPY
NASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGYLGRGPGLKTVCAARTQGGKSQK
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| BDBM301754 |
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| n/a |
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| Name | BDBM301754 |
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| Synonyms: | ((S)-6-{(R)-4-[3-Cyano-4-(3-hydroxy-3-methylbutoxy)phenoxy]-7-fluoro-indan-1-yloxy}-2,3-dihydrobenzofuran-3-yl)-acetic acid | US9597310, 44 |
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| Type | Small organic molecule |
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| Emp. Form. | C31H30FNO7 |
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| Mol. Mass. | 547.5708 |
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| SMILES | CC(C)(O)CCOc1ccc(Oc2ccc(F)c3[C@@H](CCc23)Oc2ccc3[C@H](CC(O)=O)COc3c2)cc1C#N |r| |
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| Structure | 
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