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45 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and biological evaluation of novel 2,4,5-triarylimidazole-1,2,3-triazole derivatives via click chemistry asa-glucosidase inhibitors.EBI
Jishou University
Ionic liquid-promoted multicomponent synthesis of fused tetrazolo[1,5-a]pyrimidines asa-glucosidase inhibitors.EBI
National Institute of Technology Karnataka
Inhibitory Effects of Highly Oxygenated Lanostane Derivatives from the Fungus Ganoderma lucidum on P-Glycoprotein anda-Glucosidase.EBI
Chinese Academy of Sciences
Synthesis of diethyl 4-substituted-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylates as a new series of inhibitors against yeasta-glucosidase.EBI
University of Karachi
Design, synthesis and docking study of novel tetracyclic oxindole derivatives asa-glucosidase inhibitors.EBI
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science and Technology)
Synthesis of novel indenoquinoxaline derivatives as potenta-glucosidase inhibitors.EBI
University of The Punjab
Synthesis anda-glucosidase inhibitory activity evaluation of N-substituted aminomethyl-ß-d-glucopyranosides.EBI
Xi'An Jiaotong University
(3R,4S,5R,6R,7S)-3,4,5,7-Tetrahydroxyconidine, an azetidine analogue of 6,7-diepicastanospermine and a conformationally constrained d-deoxyaltronojirimycin, from l-arabinose.EBI
University of Oxford
Mexican antidiabetic herbs: valuable sources of inhibitors ofa-glucosidases.EBI
Universidad Nacional Aut£Noma De M£Xico
Synthesis, biological activity, and molecular modeling studies of 1H-1,2,3-triazole derivatives of carbohydrates as alpha-glucosidases inhibitors.EBI
Universidade Federal Do Rio De Janeiro
Biological properties of D- and L-1-deoxyazasugars.EBI
Toyama Medical and Pharmaceutical University
Alpha-1-C-alkyl-1-deoxynojirimycin derivatives as potent and selective inhibitors of intestinal isomaltase: remarkable effect of the alkyl chain length on glycosidase inhibitory profile.EBI
Universit£
Nitrogen-in-the-ring pyranoses and furanoses: structural basis of inhibition of mammalian glycosidases.EBI
Hokuriku University
 
Potent glycosidase inhibitors, N-phenyl cyclic isourea derivatives of 5-amino- and 5-amino-1-C-(hydroxymethyl)-cyclopentane-1,2,3,4-tetraolsEBI
TBA
Towards a stable noeuromycin analog with a D-manno configuration: synthesis and glycosidase inhibition of D-manno-like tri- and tetrahydroxylated azepanes.EBI
Umr Cnrs 7201
New glucocerebrosidase inhibitors by exploration of chemical diversity of N-substituted aminocyclitols using click chemistry and in situ screening.EBI
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Selectivea-glucosidase substrates and inhibitors containing short aromatic peptidyl moieties.EBI
Seoul National University
Fluorescent-tagged sp2-iminosugars with potentß-glucosidase inhibitory activity.EBI
Universidad De Sevilla
Amplification of the inhibitory activity of miglitol by monofluorination.EBI
Martin-Luther-Universit£T Halle-Wittenberg
New polyhydroxylated pyrrolidine, piperidine, and pyrrolizidine alkaloids from Scilla sibirica.EBI
Hokuriku University
Hybrid angiogenesis inhibitors: synthesis and biological evaluation of bifunctional compounds based on 1-deoxynojirimycin and aryl-1,2,3-triazoles.EBI
University College Dublin
Synthesis of valiolamine and some precursors for bioactive carbaglycosylamines from (-)-vibo-quercitol produced by biogenesis of myo-inositol.EBI
Keio University
Aglycon specificity profiling of alpha-glucosidases using synthetic probes.EBI
Institute of Physical and Chemical Research (Riken)
Polyhydroxylated azetidine iminosugars: Synthesis, glycosidase inhibitory activity and molecular docking studies.EBI
Savitribai Phule Pune University
Pyrimidine-fused heterocycle derivatives as a novel class of inhibitors for a-glucosidase.BDB
Shiraz University
Structure-activity relationships of bergenin derivatives effect on a-glucosidase inhibition.BDB
Kinki University
Green synthesis, inhibition studies of yeast a-glucosidase and molecular docking of pyrazolylpyridazine amines.BDB
University of The Punjab
In search of new a-glucosidase inhibitors: Imidazolylpyrazole derivatives.BDB
University of The Punjab
Synthesis, molecular docking studies of hybrid benzimidazole as a-glucosidase inhibitor.BDB
Universiti Teknologi Mara (Uitm)
Design, synthesis and biological evaluation of novel coumarin thiazole derivatives as a-glucosidase inhibitors.BDB
Jishou University
Synthesis, a-glucosidase inhibitory, cytotoxicity and docking studies of 2-aryl-7-methylbenzimidazoles.BDB
Universiti Teknologi Mara (Uitm), Puncak Alam Campus
Dihydropyrano [2,3-c] pyrazole: Novel in vitro inhibitors of yeast a-glucosidase.BDB
King Abdulaziz University
Synthesis, In vitro and Docking Studies of New Flavone Ethers as a-Glucosidase Inhibitors.BDB
Universiti Teknologi Mara
Benzimidazole derivatives as new a-glucosidase inhibitors and in silico studies.BDB
Universiti Teknologi Mara (Uitm)
Pyridine sulfonamide as a small key organic molecule for the potential treatment of type-II diabetes mellitus and Alzheimer's disease: In vitro studies against yeast a-glucosidase, acetylcholinesterase and butyrylcholinesterase.BDB
Gc University
Synthesis, in vitro evaluation and molecular docking studies of biscoumarin thiourea as a new inhibitor of a-glucosidases.BDB
Universiti Teknologi Mara
Evaluation of 2-indolcarbohydrazones as potent a-glucosidase inhibitors, in silico studies and DFT based stereochemical predictions.BDB
Universiti Teknologi Mara (Uitm)
Synthesis, in vitro evaluation and molecular docking studies of thiazole derivatives as new inhibitors of a-glucosidase.BDB
Hazara University
Isatin based Schiff bases as inhibitors of a-glucosidase: Synthesis, characterization, in vitro evaluation and molecular docking studies.BDB
Hazara University
Triazinoindole analogs as potent inhibitors of a-glucosidase: synthesis, biological evaluation and molecular docking studies.BDB
Hazara University
Organocatalyzed solvent free an efficient novel synthesis of 2,4,5-trisubstituted imidazoles for a-glucosidase inhibition to treat diabetes.BDB
Comsats Institute of Information Technology
Novel synthesis of dihydropyrimidines for a-glucosidase inhibition to treat type 2 diabetes: in vitro biological evaluation and in silico docking.BDB
Comsats Institute of Information Technology
New insights into the pharmacological chaperone activity of c2-substituted glucoimidazoles for the treatment of Gaucher disease.BDB
Nankai University
Antioxidant, a-glucosidase and xanthine oxidase inhibitory activity of bioactive compounds from maize (Zea mays L.).BDB
Srtm University
A novel competitive class of α-glucosidase inhibitors: (E)-1-phenyl-3-(4-styrylphenyl)urea derivatives.BDB
Gyeongsang National University