null
SMILES Cl.COc1ccc(\C=C\C2=NN(CCCCN)C(=O)N(Cc3ccc(cc3)-c3ccccc3)c3ccccc23)cc1
InChI Key InChIKey=HMFTXUPXTQWPNX-OQKWZONESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50269946
Affinity DataEC50: 3.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 1.74E+3nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced G12 activation by measuring URP pEC50...More data for this Ligand-Target Pair
Affinity DataEC50: 7.10nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced Gq activation by measuring URP pEC50 ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.24E+3nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced G12 activation by measu...More data for this Ligand-Target Pair
Affinity DataEC50: 8.5nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced Gq activation by measur...More data for this Ligand-Target Pair