null
SMILES Cc1ccc(cc1)-c1c(\C=C\C#N)n(CCCO)c2ncnc(N)c12
InChI Key InChIKey=LPADWFDQODOOMS-DUXPYHPUSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 259803
TargetRibosomal protein S6 kinase alpha-3 [399-740](Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA
US Patent
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA
US Patent
Affinity DataIC50: 750nMpH: 8.0 T: 2°CAssay Description:RSK2 CTD and His6-ERK2 were expressed and purified as described (Cohen et al., Science, 308: 1318). The C436V mutant of RSK2 CTD was generated by Qui...More data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
University of Pittsburgh
Curated by ChEMBL
University of Pittsburgh
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of RSK2 in human MDA-MB-231 cells after 2 hrsMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3 [399-740,C436V](Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA
US Patent
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA
US Patent
Affinity DataIC50: 1.50E+3nMpH: 8.0 T: 2°CAssay Description:RSK2 CTD and His6-ERK2 were expressed and purified as described (Cohen et al., Science, 308: 1318). The C436V mutant of RSK2 CTD was generated by Qui...More data for this Ligand-Target Pair