null

SMILES Nc1ncc(cc1-c1cc2cc(NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)ccc2s1)-c1nnn(CCCO)n1

InChI Key InChIKey=HSVUTNRAXRQFMN-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 308056   

TargetInterferon-induced, double-stranded RNA-activated protein kinase(Homo sapiens (Human))
ALLERGAN, INC.

US Patent
LigandPNGBDBM308056(US10011593, Ex. 6 | US9650366, 6)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Biochemical PDGFRβ kinase assays were performed in 96 well microtiter plates that were coated overnight with 75 μg of poly-Glu-Tyr (4:1) in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QN68VGUS Patent
TargetInterferon-induced, double-stranded RNA-activated protein kinase(Homo sapiens (Human))
ALLERGAN, INC.

US Patent
LigandPNGBDBM308056(US10011593, Ex. 6 | US9650366, 6)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24J0HGVUS Patent