null
SMILES CSCC[C@@H](NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)[C@@H](C)NC(=O)[C@@H](CCC(O)=O)NC(=O)[C@@H](CCC(O)=O)NC(=O)[C@@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@@H](N)CCC(O)=O)C(=O)N[C@H](CC(O)=O)C(=O)N[C@H](Cc1ccccc1)C(N)=O
InChI Key InChIKey=AOXOCDRNSPFDPE-UKEONUMOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50026690
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for in vitro inhibition of the binding of [125I]-(Nle11)-HG-13 to Histamine H2 receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
NCI-Frederick Cancer Research and Development Center
Curated by ChEMBL
NCI-Frederick Cancer Research and Development Center
Curated by ChEMBL
Affinity DataKd: 3.20nMAssay Description:Tested in vitro for gastrin binding to gastrin receptors from guinea pig gastric glandsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
NCI-Frederick Cancer Research and Development Center
Curated by ChEMBL
NCI-Frederick Cancer Research and Development Center
Curated by ChEMBL
Affinity DataKd: 1.40nMAssay Description:Tested in vitro by the gastrin binding assay for the competitive binding with iodinated gastrin for the gastrin receptors in AR42J cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
NCI-Frederick Cancer Research and Development Center
Curated by ChEMBL
NCI-Frederick Cancer Research and Development Center
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair