null
SMILES Clc1cc(Oc2ccccn2)cc(c1)N1Cc2ccccc2S1(=O)=O
InChI Key InChIKey=ROJVYIHWPWITEK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50196402
TargetFree fatty acid receptor 4(Homo sapiens (Human))
University of Southern Denmark
Curated by ChEMBL
University of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Agonist activity at C-terminal YFP-tagged human FFA4 expressed in HEK293 cells in presence of coelentrazine h by BRET based beta-arrestin-2 interacti...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
University of Southern Denmark
Curated by ChEMBL
University of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at human FFA4 expressed in human Flp-In T-REx293 cells by Fura2-AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University of Southern Denmark
Curated by ChEMBL
University of Southern Denmark
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity against human FFA1 expressed in human Flp-In T-REx293 cells assessed as as reduction in TUG770-induced response by Fura2-AM dye b...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
University of Southern Denmark
Curated by ChEMBL
University of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Agonist activity at C-terminal YFP-tagged human FFA4 expressed in HEK293 cells in presence of coelentrazine h by BRET based beta-arrestin-2 interacti...More data for this Ligand-Target Pair
Affinity DataEC50: 72nMAssay Description:Agonist activity mouse FFA4 by Gq-dependent calcium mobilization assayMore data for this Ligand-Target Pair