null
SMILES COc1cc(ccc1N)-c1cnc2c(snc2c1)N1C[C@H](C)O[C@H](C)C1
InChI Key InChIKey=VOFMQYIALBSDFI-TXEJJXNPSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50288800
Affinity DataKd: 89nMAssay Description:Binding affinity to DNA-tagged human GAK expressed in Escherichia coli BL21 using immobilised ligand incubated for 1 hr by quantitative PCRMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Inhibition of wild-type human partial length KIT (I571 to D952 residues) expressed in bacterial expression system by ATP-site competition binding ass...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair