null
SMILES CCOc1ccc(Cc2cc([C@@H]3S[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(OC)cc2C)cc1
InChI Key InChIKey=WHSOLWOTCHFFBK-ZQGJOIPISA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50315426
Affinity DataKi: 1.10nMAssay Description:Competitive inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-alpha-methylglucoside uptakeMore data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition of human SGLT1 expressed in CHOK1 cells assessed as inhibition of glucose uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of SGLT2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Inhibition of SGLT2 (unknown origin)More data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition of human SGLT1More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition OF SGLT2 (unknown origin)More data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Inhibition of SGLT1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human SGLT2 expressed in CHOK1 cells assessed as inhibition of glucose uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair