null
SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2ccc(F)cc2)c1=O
InChI Key InChIKey=QUIIIYITNGOFEI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50384774
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
The Regents of The University of Michigan; The University of Bath
US Patent
The Regents of The University of Michigan; The University of Bath
US Patent
Affinity DataIC50: 30nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
The Regents of The University of Michigan; The University of Bath
US Patent
The Regents of The University of Michigan; The University of Bath
US Patent
Affinity DataIC50: 1.10E+4nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
TargetRegulator of G-protein signaling 16(Homo sapiens (Human))
The Regents of The University of Michigan; The University of Bath
US Patent
The Regents of The University of Michigan; The University of Bath
US Patent
Affinity DataIC50: 3.50E+3nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In DepthDetails
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
The Regents of The University of Michigan; The University of Bath
US Patent
The Regents of The University of Michigan; The University of Bath
US Patent
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
The Regents of The University of Michigan; The University of Bath
US Patent
The Regents of The University of Michigan; The University of Bath
US Patent
Affinity DataIC50: 30nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
TargetRegulator of G-protein signaling 19(Homo sapiens (Human))
The Regents of The University of Michigan; The University of Bath
US Patent
The Regents of The University of Michigan; The University of Bath
US Patent
Affinity DataIC50: 120nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair