null
SMILES [H][C@@]12Oc3c4c(C[C@@]5([H])N(CC6CC6)CC[C@@]14[C@@]5(O)CC[C@H]2NC(=O)c1cnc[nH]1)ccc3O
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50586081
Affinity DataKi: 0.580nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cells in presence of naltrexone incubated for 1.5 hrs by competitive radioligand bindin...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to mouse kappa opioid receptor expressed in CHO cells in presence of U50488 incubated for 1.5 hrs by competitive radioligand binding...More data for this Ligand-Target Pair
Affinity DataKi: 209nMAssay Description:Binding affinity to human delta opioid receptor in presence of SNC80 incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Antagonist activity at mouse mu opioid receptor expressed in CHO cell membrane assessed as reduction in DAMGO-induced [3S]-GTPgammaS binding incubate...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Antagonist activity at kappa opioid receptor (unknown origin) expressed in CHO cell membrane assessed as reduction in U50,488H-induced [3S]-GTPgammaS...More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Antagonist activity at human delta opioid receptor expressed in CHO cell membrane assessed as reduction in SNC80-induced [3S]-GTPgammaS binding incub...More data for this Ligand-Target Pair