Compile Data Set for Download or QSAR
Found 112 Enz. Inhib. hit(s) with Target = 'Histone lysine demethylase PHF8'
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276050(2-[1-(3,4-dihydro-2H-chromen-4-ylmethyl)imidazol-4...)copy SMILES
Affinity DataIC50: 100nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276044(2-[1-[2-(2-chlorophenyl)ethyl]imidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276067(2-[1-[(3-chloro-2-fluorophenyl)methyl]imidazol-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM50155508(CHEMBL3780833)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8GC9PubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM50155507(CHEMBL3780904)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8GC9PubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM50155505(CHEMBL3781414)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8GC9PubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM50155449(CHEMBL3780958)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8GC9PubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM50155450(CHEMBL3779953)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8GC9PubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM50155509(CHEMBL3780689)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8GC9PubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276082(1-benzyl-4-{1H-[1,2,3]triazolo[4,5-c]pyridin-6-yl}...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276053(4-[2-[1-(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)i...)copy SMILES
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276054(4-[2-[1-(2-naphthalen-1-ylethyl)imidazol-4-yl]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276057(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276058(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276059(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276060(2-[1-[[2-chloro-3-(trifluoromethyl)phenyl]methyl]i...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276061(2-[1-(2-naphthalen-1-ylethyl)imidazol-4-yl]-4-(1H-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276062(2-[5-(4-fluoro-3-methoxyphenyl)-1-methylimidazol-4...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276066(2-[1-[(2-fluoro-3-methylphenyl)methyl]imidazol-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276048(4-(1H-triazol-4-yl)-2-[1-[2-[2-(2,2,2-trifluoroeth...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276047(2-[1-[2-(2-ethoxyphenyl)ethyl]imidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276046(2-[1-(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)imid...)copy SMILES
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276045(2-[1-[2-(2-methoxyphenyl)ethyl]imidazol-4-yl]-4-(1...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276043(2-[1-(1-phenylethyl)imidazol-4-yl]-4-(1H-triazol-4...)copy SMILES
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276041(2-[5-(4-fluorophenyl)-1-methylimidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276040(2-[1-[(2-chlorophenyl)methyl]imidazol-4-yl]-4-(1H-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276039(2-(1-methylimidazol-4-yl)-4-(1H-triazol-4-yl)pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276093(2-(5-bromo-1-(2-chlorobenzyl)-1H-imidazol-4-yl)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276049(2-[1-[2-[2-(cyclopropylmethoxy)phenyl]ethyl]imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276068(2-[1-[(2-fluoro-3-methoxyphenyl)methyl]imidazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276069(4-(1H-triazol-4-yl)-2-[1-[2-[2-(trifluoromethyl)ph...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276070(2-[1-[2-(2-chlorophenyl)-2-methylpropyl]imidazol-4...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276072(4-(1H-triazol-4-yl)-2-[1-[2-[2-(trifluoromethoxy)p...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276073(4-(5-fluoro-1H-triazol-4-yl)-2-[1-(2-naphthalen-1-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM50395083(CHEMBL2164246)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276042(2-[5-[2-(cyclopropylmethoxy)-4-fluorophenyl]-1-met...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276051(4-[2-[1-[(2-chlorophenyl)methyl]imidazol-4-yl]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276052(4-[2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276055(2-[1-[2-(2-phenylmethoxyphenyl)ethyl]imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276056(2-[1-[2-(2-phenoxyphenyl)ethyl]imidazol-4-yl]-4-(1...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276063(2-[5-(3-ethoxy-4-fluorophenyl)-1-methylimidazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276064(2-[1-[[2-fluoro-3-(trifluoromethoxy)phenyl]methyl]...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276065(2-[1-[2-(2-phenylphenyl)ethyl]imidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276071(2-[1-(1-phenylpropan-2-yl)imidazol-4-yl]-4-(1H-tri...)copy SMILES
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276074(4-(5-chloro-1H-triazol-4-yl)-2-[1-(2-naphthalen-1-...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM373122(4-[2-[5-2-cyclopropylmethoxy)-4- fluorophenyl]-1-m...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276079(2-[5-[2-(cyclopropylmethoxy)-4-fluorophenyl]-1-met...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276080(1-(cyclopropylmethyl)-4-{1H-[1,2,3]triazolo[4,5-c]...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276081(4-{1H-[1,2,3]triazolo[4,5-c]pyridin-6-yl}-1-(2,2,2...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
GSK

LigandPNGBDBM276083(1-[(2-chlorophenyl)methyl]-4-{1H-[1,2,3]triazolo[4...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FT8PBQUS Patent
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