Compile Data Set for Download or QSAR
Found 44 Enz. Inhib. hit(s) with Target = 'Phospholipase A-2-activating protein'
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50042034((5Z)-7-Oxozeaenol | 5Z-7-Oxozeaenol | CHEBI:67559 ...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of TNFalpha-PLAP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8H9TPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50245461(CHEMBL4068569)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of TNFalpha-PLAP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8H9TPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41890(2-(1-benzimidazolyl)-1-(3,4-dihydroxyphenyl)ethano...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41891(1-(3,4-dihydroxyphenyl)-2-(2-methyl-1-benzimidazol...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41891(1-(3,4-dihydroxyphenyl)-2-(2-methyl-1-benzimidazol...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50237956(1-(3,4-dihydroxyphenyl)-2-(1-(4-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41887(1-(3,4-dihydroxyphenyl)-2-(1-imidazolyl)ethanone;h...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309563(2-(2-(3,4-dihydroxyphenyl)-2-oxoethylthio)-4-(meth...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309564(1-(3,4-dihydroxyphenyl)-2-(4,6-dimethylpyrimidin-2...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309565(1-(3,4-dihydroxyphenyl)-2-(4-methyl-1H-pyrazol-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309567(3-(2-(3,4-dihydroxyphenyl)-2-oxoethyl)-6,7-dimetho...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41889(1-(3,4-dihydroxyphenyl)-2-(2-methyl-1-imidazolyl)e...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41889(1-(3,4-dihydroxyphenyl)-2-(2-methyl-1-imidazolyl)e...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41888(1-(3,4-dihydroxyphenyl)-2-(2-ethyl-1-imidazolyl)et...)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM41888(1-(3,4-dihydroxyphenyl)-2-(2-ethyl-1-imidazolyl)et...)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46047(1-[3,4-bis(oxidanyl)phenyl]-2-(4-bromanyl-2-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309588(CHEMBL589752 | L-homoarginine)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM18073((2S)-2-amino-3-phenylpropanoic acid | CHEMBL301523...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM10847(1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dion...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50241179((S)-6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiaz...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM21974((2S)-2-amino-3-(1H-indol-3-yl)propanoic acid | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50219348((2S)-2-amino-4-methylpentanoic acid | (S)-(+)-leuc...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309587(CHEMBL598548 | L-leucinamide | LEUCINE AMIDE)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46053(1-(3,4-dihydroxyphenyl)-2-(4-methyl-1-imidazolyl)e...)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46052(1-(3,4-dihydroxyphenyl)-2-(5,6-dimethyl-1-benzimid...)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309570(1-(3,4-dihydroxyphenyl)-2-(4-methyl-5-phenyl-4H-1,...)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46050(2-(1H-benzimidazol-2-ylamino)-1-(3,4-dihydroxyphen...)copy SMILEScopy InChI
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50245475(CHEMBL4103122)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TNFalpha-PLAP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8H9TPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50245474(CHEMBL4078847)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TNFalpha-PLAP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8H9TPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46051(1-(3,4-dihydroxyphenyl)-2-(1,2,4-triazol-4-yl)etha...)copy SMILEScopy InChI
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46048(1-[3,4-bis(oxidanyl)phenyl]-2-(4-bromanylimidazol-...)copy SMILEScopy InChI
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46049(1-(3,4-dihydroxyphenyl)-2-(2-phenyl-1-imidazolyl)e...)copy SMILEScopy InChI
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46041(1-(3,4-dihydroxyphenyl)-2-(isopropylamino)ethanone...)copy SMILEScopy InChI
Affinity DataIC50: 3.93E+4nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309578(4-((4,6-dimethylpyrimidin-2-ylamino)methyl)benzene...)copy SMILEScopy InChI
Affinity DataIC50: 5.12E+4nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309580(2-(4,6-dimethylpyrimidin-2-ylthio)-1-(3-hydroxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309579(2-(4,6-dimethylpyrimidin-2-ylthio)-1-(4-hydroxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50299523(2,5-Dimethoxy-N-(quinolin-3-yl)benzenesulfonamide ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by luminescent assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8T9MPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309585(CHEMBL599678 | N-(3,4-dihydroxyphenethyl)-4,5-dime...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46046(2-(4,6-dimethylpyrimidin-2-yl)sulfanyl-1-(3-methox...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM46045(1-(1,3-benzodioxol-5-yl)-2-(4,6-dimethylpyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309583(2-(4,6-dimethylpyrimidin-2-ylthio)-1-(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309584(CHEMBL599476 | N-(3,4-dihydroxybenzyl)-4,5-dimethy...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM32012(1-(3,4-Dihydroxy-phenyl)-2-(5-phenyl-4H-[1,2,4]tri...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed
TargetPhospholipase A-2-activating protein(Homo sapiens (Human))
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50309586(2-(5-(3-aminophenyl)-4-methyl-4H-1,2,4-triazol-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PLAP by analogous luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JHRPubMed