Compile Data Set for Download or QSAR
Found 55 Enz. Inhib. hit(s) with Target = 'Isoform 2 of Histone lysine demethylase PHF8 (2)'
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276050(2-[1-(3,4-dihydro-2H-chromen-4-ylmethyl)imidazol-4...)copy SMILES
Affinity DataIC50: 100nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276067(2-[1-[(3-chloro-2-fluorophenyl)methyl]imidazol-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 100nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276044(2-[1-[2-(2-chlorophenyl)ethyl]imidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 100nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276043(2-[1-(1-phenylethyl)imidazol-4-yl]-4-(1H-triazol-4...)copy SMILES
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276045(2-[1-[2-(2-methoxyphenyl)ethyl]imidazol-4-yl]-4-(1...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276046(2-[1-(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)imid...)copy SMILES
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276047(2-[1-[2-(2-ethoxyphenyl)ethyl]imidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276048(4-(1H-triazol-4-yl)-2-[1-[2-[2-(2,2,2-trifluoroeth...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276049(2-[1-[2-[2-(cyclopropylmethoxy)phenyl]ethyl]imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276041(2-[5-(4-fluorophenyl)-1-methylimidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276093(2-(5-bromo-1-(2-chlorobenzyl)-1H-imidazol-4-yl)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276039(2-(1-methylimidazol-4-yl)-4-(1H-triazol-4-yl)pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276040(2-[1-[(2-chlorophenyl)methyl]imidazol-4-yl]-4-(1H-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276082(1-benzyl-4-{1H-[1,2,3]triazolo[4,5-c]pyridin-6-yl}...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276073(4-(5-fluoro-1H-triazol-4-yl)-2-[1-(2-naphthalen-1-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276072(4-(1H-triazol-4-yl)-2-[1-[2-[2-(trifluoromethoxy)p...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276070(2-[1-[2-(2-chlorophenyl)-2-methylpropyl]imidazol-4...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276069(4-(1H-triazol-4-yl)-2-[1-[2-[2-(trifluoromethyl)ph...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276068(2-[1-[(2-fluoro-3-methoxyphenyl)methyl]imidazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276066(2-[1-[(2-fluoro-3-methylphenyl)methyl]imidazol-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276062(2-[5-(4-fluoro-3-methoxyphenyl)-1-methylimidazol-4...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276061(2-[1-(2-naphthalen-1-ylethyl)imidazol-4-yl]-4-(1H-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276060(2-[1-[[2-chloro-3-(trifluoromethyl)phenyl]methyl]i...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276059(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276058(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276057(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276054(4-[2-[1-(2-naphthalen-1-ylethyl)imidazol-4-yl]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276053(4-[2-[1-(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)i...)copy SMILES
Affinity DataIC50: 550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276042(2-[5-[2-(cyclopropylmethoxy)-4-fluorophenyl]-1-met...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276051(4-[2-[1-[(2-chlorophenyl)methyl]imidazol-4-yl]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276088(1-(2-chlorophenyl)-4-{1H-[1,2,3]triazolo[4,5-c]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276089(1-(3-chlorophenyl)-4-{1H-[1,2,3]triazolo[4,5-c]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276071(2-[1-(1-phenylpropan-2-yl)imidazol-4-yl]-4-(1H-tri...)copy SMILES
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276090(1-(3,5-dichlorophenyl)-4-{1H-[1,2,3]triazolo[4,5-c...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276091(5-(4-fluorophenyl)-1-methyl-4-{1H-[1,2,3]triazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276074(4-(5-chloro-1H-triazol-4-yl)-2-[1-(2-naphthalen-1-...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276087(1-(4-chlorophenyl)-4-{1H-[1,2,3]triazolo[4,5-c]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276052(4-[2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276079(2-[5-[2-(cyclopropylmethoxy)-4-fluorophenyl]-1-met...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276077(4-[2-[5-[2-(cyclopropylmethoxy)-4-fluorophenyl]-1-...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276086(1-[(3,4-dichlorophenyl)methyl]-4-{1H-[1,2,3]triazo...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276065(2-[1-[2-(2-phenylphenyl)ethyl]imidazol-4-yl]-4-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276064(2-[1-[[2-fluoro-3-(trifluoromethoxy)phenyl]methyl]...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276063(2-[5-(3-ethoxy-4-fluorophenyl)-1-methylimidazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276085(1-[(4-chlorophenyl)methyl]-4-{1H-[1,2,3]triazolo[4...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276084(1-[(3-chlorophenyl)methyl]-4-{1H-[1,2,3]triazolo[4...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276083(1-[(2-chlorophenyl)methyl]-4-{1H-[1,2,3]triazolo[4...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276092(5-[2-(cyclopropylmethoxy)-4-fluorophenyl]-1-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276081(4-{1H-[1,2,3]triazolo[4,5-c]pyridin-6-yl}-1-(2,2,2...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
TargetIsoform 2 of Histone lysine demethylase PHF8 (2)(Homo sapiens (Human))
Celgene Quanticel Research, Inc.

US Patent
LigandPNGBDBM276080(1-(cyclopropylmethyl)-4-{1H-[1,2,3]triazolo[4,5-c]...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7X0XUS Patent
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