Compile Data Set for Download or QSAR
Found 196 with Last Name = 'heitz' and Initial = 'a'
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50005601(CHEMBL2369819)copy SMILEScopy InChI
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50408923(CHEMBL2114155)copy SMILEScopy InChI
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089280(CHEMBL437655 | JMV 1535)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089284(CHEMBL265856 | JMV 1803)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089285(CHEMBL415110 | JMV 1799)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089282((D)Phe-Gln-Trp-Ala-Val-Gly-His-Leu-Leu-NH2 | CHEMB...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089281(CHEMBL386480 | JMV 1802)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089291(CHEMBL415021 | JMV 1813)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089278(CHEMBL411016 | JMV 1801)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089279(CHEMBL406013 | JMV 1719)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089286(CHEMBL407022 | JMV 1693)copy SMILEScopy InChI
Affinity DataKi:  127nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50408922(CHEMBL2115179)copy SMILEScopy InChI
Affinity DataKi:  225nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089288(Bombesin analogues | CHEMBL415022)copy SMILEScopy InChI
Affinity DataKi:  300nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089292(Bombesin analogues | CHEMBL439440)copy SMILEScopy InChI
Affinity DataKi:  500nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089290(Bombesin analogues | CHEMBL413938)copy SMILEScopy InChI
Affinity DataKi:  650nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089293(Bombesin analogues | CHEMBL407481)copy SMILEScopy InChI
Affinity DataKi:  2.25E+3nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089287(Bombesin analogues | CHEMBL384242)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGastrin-releasing peptide receptor(RAT)
CNRS-Universités Montpellier I & II

Curated by ChEMBL
LigandPNGBDBM50089289(Bombesin analogues | CHEMBL384241)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J990KPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19331(CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nM EC50:  3nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50366689(GHRELIN)copy SMILEScopy InChI
Affinity DataIC50: 0.390nMAssay Description:Binding affinity towards cloned human Growth hormone secretagogue receptor type I in LLC PK-1 cells using [125I][His9]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40NJPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19333(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nM EC50:  0.600nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19332(N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nM EC50:  1.60nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)copy SMILEScopy InChI
Affinity DataIC50: 0.760nMAssay Description:Binding affinity towards cloned human Growth hormone secretagogue receptor type I in LLC PK-1 cells using [125I][His9]-ghrelin as radioligandMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19334(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-(2-ph...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nM EC50:  6.10nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50125888(CHEMBL282891 | Piperidine-4-carboxylic acid [1-[(R...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Binding affinity towards cloned human Growth hormone secretagogue receptor type I in LLC PK-1 cells using [125I][His9]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40NJPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19312((2S)-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nM Kd:  11nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19294(2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19349(N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...)copy SMILEScopy InChI
Affinity DataIC50: 6nM Kd:  51nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19294(2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...)copy SMILEScopy InChI
Affinity DataIC50: 6nM Kd:  4nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19318(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1...)copy SMILEScopy InChI
Affinity DataIC50: 6.5nM EC50:  5.30nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19323((3R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 7nM EC50:  36nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19308((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataIC50: 9nM Kd:  6nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19310((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 9.5nM Kd:  13nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50366689(GHRELIN)copy SMILEScopy InChI
Affinity DataIC50: 9.80nMAssay Description:Binding affinity towards human pituitary Growth hormone secretagogue receptor using [125I][Tyr4]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40NJPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19321((3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataIC50: 10nM EC50:  2.5nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50208662((R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19326((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 11nM Kd:  27nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50208646((R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-phenethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50125889(CHEMBL214233 | Tyr-Ala-hexarelin)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Binding affinity towards human pituitary Growth hormone secretagogue receptor using [125I][Tyr4]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40NJPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50208678((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19319(N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-...)copy SMILEScopy InChI
Affinity DataIC50: 13nM EC50:  9.90nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50208670((R)-N-(1-(4-(2-(1H-indol-3-yl)ethyl)-5-(3-(1H-indo...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19293((R)-N-(1-(5-(2-(1H-Indol-3-yl)ethyl)-4-benzyl-4H-1...)copy SMILEScopy InChI
Affinity DataIC50: 15nM EC50:  64nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19293((R)-N-(1-(5-(2-(1H-Indol-3-yl)ethyl)-4-benzyl-4H-1...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19322((3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 16nM Kd:  10nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50125877(CHEMBL281173 | [(S)-1-[(R)-2-(2-Amino-2-methyl-pro...)copy SMILEScopy InChI
Affinity DataIC50: 16.2nMAssay Description:Binding affinity towards human pituitary Growth hormone secretagogue receptor using [125I][Tyr4]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40NJPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50125881(2-Amino-N-[1-[(R)-(S)-1-(3-ethyl-ureido)-2-(1H-ind...)copy SMILEScopy InChI
Affinity DataIC50: 16.9nMAssay Description:Binding affinity towards human pituitary Growth hormone secretagogue receptor using [125I][Tyr4]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40NJPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50208689((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxyb...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Displacement of [125I-His9]ghrelin from human GHS1a receptor expressed in LLC PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251HW6PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Binding affinity towards human pituitary Growth hormone secretagogue receptor using [125I][Tyr4]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40NJPubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19344(N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)e...)copy SMILEScopy InChI
Affinity DataIC50: 18nM EC50:  8.70nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
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