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Found 117 with Last Name = 'folkes' and Initial = 'aj'
LigandPNGBDBM50363990(CHEMBL1949915)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347087(CHEMBL1796273)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347090(CHEMBL1796276)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419754(CHEMBL1949910)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419769(CHEMBL1950034)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419759(CHEMBL1949916)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419770(CHEMBL1950035)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419761(CHEMBL1949919)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347076(CHEMBL1796761)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419760(CHEMBL1949918)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419758(CHEMBL1949914)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419773(CHEMBL1949917)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419762(CHEMBL1949920)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419771(CHEMBL1950036)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50363991(CHEMBL1796763)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419765(CHEMBL1949923)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419766(CHEMBL1949924)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419764(CHEMBL1949922)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419772(CHEMBL1950037)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419757(CHEMBL1949913)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419757(CHEMBL1949913)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419756(CHEMBL1949912)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419763(CHEMBL1949921)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347085(CHEMBL1796271)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419758(CHEMBL1949914)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347076(CHEMBL1796761)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419768(CHEMBL1949926)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50363990(CHEMBL1949915)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419769(CHEMBL1950034)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419767(CHEMBL1949925)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419766(CHEMBL1949924)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419765(CHEMBL1949923)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419773(CHEMBL1949917)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419756(CHEMBL1949912)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419759(CHEMBL1949916)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419761(CHEMBL1949919)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419755(CHEMBL1949911)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419774(CHEMBL1950038)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419764(CHEMBL1949922)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419770(CHEMBL1950035)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419754(CHEMBL1949910)copy SMILEScopy InChI
Affinity DataKi:  69nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347090(CHEMBL1796276)copy SMILEScopy InChI
Affinity DataKi:  87nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419760(CHEMBL1949918)copy SMILEScopy InChI
Affinity DataKi:  108nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347087(CHEMBL1796273)copy SMILEScopy InChI
Affinity DataKi:  114nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419771(CHEMBL1950036)copy SMILEScopy InChI
Affinity DataKi:  144nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419772(CHEMBL1950037)copy SMILEScopy InChI
Affinity DataKi:  199nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50363991(CHEMBL1796763)copy SMILEScopy InChI
Affinity DataKi:  204nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50419762(CHEMBL1949920)copy SMILEScopy InChI
Affinity DataKi:  247nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347085(CHEMBL1796271)copy SMILEScopy InChI
Affinity DataKi:  272nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Piramed Pharma

LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)copy SMILEScopy InChI
Affinity DataKi:  580nM ΔG°:  -35.6kJ/molepH: 7.5 T: 2°CAssay Description:Mammalian target of rapamycin (mTOR) was assayed by monitoring phosphorylation of GFP-4EBP using a homogeneous time-resolved fluorescence resonance e...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222S23PubMed
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