Compile Data Set for Download or QSAR
Found 53 with Last Name = 'casagrande' and Initial = 'as'
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 0.220nMAssay Description:Inhibition of human DYRK1A using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 0.220nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:Inhibition of human DYRK1A using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 0.590nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 0.590nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434352(CHEMBL2386748 | US9446044, 78)copy SMILEScopy InChI
Affinity DataIC50: 0.940nMAssay Description:Inhibition of human DYRK1A using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434364(CHEMBL2386764 | US9446044, 65)copy SMILEScopy InChI
Affinity DataIC50: 0.980nMAssay Description:Inhibition of human DYRK1A using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246384(US9446044, 71)copy SMILEScopy InChI
Affinity DataIC50: 0.990nMAssay Description:Inhibition of human DYRK1A using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434352(CHEMBL2386748 | US9446044, 78)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246384(US9446044, 71)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434364(CHEMBL2386764 | US9446044, 65)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of DYRK2 (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 7.40nMAssay Description:Inhibition of GSK3A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human DYRK1A using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))TBA
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Inhibition of GSK3A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))TBA
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK2 (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of DYRK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human DYRK1A using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))TBA
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))TBA
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))TBA
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Inhibition of DYRK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))TBA
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 143nMAssay Description:Inhibition of GSK3B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))TBA
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 221nMAssay Description:Inhibition of GSK3B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))TBA
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of CLK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
LigandPNGBDBM246383(US9446044, 69)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of DYRK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))TBA
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CLK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561942(CHEMBL4762738)copy SMILES
Affinity DataEC50:  157nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561943(CHEMBL4792864)copy SMILES
Affinity DataEC50:  530nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561944(CHEMBL4796139)copy SMILES
Affinity DataEC50:  309nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561945(CHEMBL4760298)copy SMILES
Affinity DataEC50:  4.17E+3nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561946(CHEMBL4759170)copy SMILES
Affinity DataEC50:  5.90E+3nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561947(CHEMBL4756278)copy SMILES
Affinity DataEC50: >5.00E+4nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561948(CHEMBL4755690)copy SMILES
Affinity DataEC50:  510nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561949(CHEMBL4798692)copy SMILES
Affinity DataEC50:  677nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561950(CHEMBL4784420)copy SMILES
Affinity DataEC50:  500nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561951(CHEMBL4793431)copy SMILES
Affinity DataEC50:  1.90E+3nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561952(CHEMBL4791976)copy SMILES
Affinity DataEC50: >5.00E+4nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561941(CHEMBL4791949)copy SMILES
Affinity DataEC50:  580nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561940(CHEMBL4791999)copy SMILES
Affinity DataEC50:  890nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50561939(CHEMBL4758550)copy SMILES
Affinity DataEC50:  1.26E+3nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
TargetUtrophin(Homo sapiens)TBA
LigandPNGBDBM50542765(CHEMBL4638592)copy SMILEScopy InChI
Affinity DataEC50:  244nMAssay Description:Modulation of human utrophinA expressed in mouse H2K-mdx utrnA-luc cells assessed as upregulation of utrophin production after 24 hrs by luciferase r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23200M9PubMed
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