TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 0.170nMAssay Description:Evaluated for binding activity against [3H]ketanserin as radioligand for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Compound was evaluated for binding activity against [3H]pyrilamine as radioligand for Histamine H1 receptorMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 5.5nMAssay Description:Compound was evaluated for binding activity against [3H]-WB- 4101 as radioligand for alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 164nMAssay Description:Compound was evaluated for binding activity against [3H]-haloperidol as radioligand for Dopamine receptor D2More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 4.42E+3nMAssay Description:Compound was evaluated for binding activity against [3H]haloperidol as radioligand for Dopamine receptor D2More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Affinity DataIC50: 0.562nMAssay Description:Evaluated for binding activity against [3H]ketanserin as radioligand for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Compound was evaluated for binding activity against [3H]pyrilamine as radioligand for Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for binding activity against [3H]pyrilamine as radioligand for Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 417nMAssay Description:Compound was evaluated for binding activity against [3H]haloperidol as radioligand for Dopamine receptor D2More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for binding activity against [3H]sufentanil opiate receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for binding activity against [3H]clonidine as radioligand for alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for binding activity against [3H]dexetimide as radioligand for muscarinic-acetylcholine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for binding activity against [3H]dihydroalprenolol as radioligand for beta adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+3nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of interaction between GST-tagged Bcl-xl and Bak by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.62E+3nMAssay Description:Compound was evaluated for binding activity against [3H]-5-HT as radioligand for serotonin S1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.91E+3nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of interaction between GST-tagged Bcl-xl and Bak by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of interaction between GST-tagged Bcl-xl and Bak by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.29E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
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