Compile Data Set for Download or QSAR
Found 210 with Last Name = 'scudiero' and Initial = 'd'
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of RSK2 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of RSK1 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of CHK1 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Aurora A using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence micropl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.830nMAssay Description:Inhibition of c-Src using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of LCK using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of c-Src using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMedDrugBank
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of LCK using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate a...More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of ALK using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of CHK2 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 8.60nMAssay Description:Inhibition of ZAP70 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Inhibition of LCK using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of CHK2 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of ALK using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Inhibition of CHK1 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 80nMpH: 7.5 T: 2°CAssay Description:NSC 109555 was diluted in water. All other drugs were dissolved in DMSO, in which case the final DMSO concentration in reactions was 10%, and the con...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67F9QPubMed
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)copy SMILEScopy InChI
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:NSC 109555 was diluted in water. All other drugs were dissolved in DMSO, in which case the final DMSO concentration in reactions was 10%, and the con...More data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 131nMAssay Description:Inhibition of RSK1 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 153nMAssay Description:Inhibition of c-Src using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 184nMAssay Description:Inhibition of RSK2 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
LigandPNGBDBM34063(DDUG | NSC 109555 | diacetyldiphenylurea bisguanyl...)copy SMILEScopy InChI
Affinity DataIC50: 200nMpH: 7.2 T: 2°CAssay Description:The IMAP Screening Express Kit (Molecular Devices, Sunnyvale, CA) was used for the high-throughput screening experiments. Compounds from the Developm...More data for this Ligand-Target Pair
LigandPNGBDBM34063(DDUG | NSC 109555 | diacetyldiphenylurea bisguanyl...)copy SMILEScopy InChI
Affinity DataIC50: 240nMpH: 7.5 T: 2°CAssay Description:NSC 109555 was diluted in water. All other drugs were dissolved in DMSO, in which case the final DMSO concentration in reactions was 10%, and the con...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 405nMAssay Description:Inhibition of c-Met using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
LigandPNGBDBM16591((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 420nMpH: 7.5 T: 2°CAssay Description:NSC 109555 was diluted in water. All other drugs were dissolved in DMSO, in which case the final DMSO concentration in reactions was 10%, and the con...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67F9QPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355550(CHEMBL1910608)copy SMILEScopy InChI
Affinity DataIC50: 607nMAssay Description:Inhibition of RSK2 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355557(CHEMBL1910625)copy SMILEScopy InChI
Affinity DataIC50: 970nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355550(CHEMBL1910608)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of RSK1 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355550(CHEMBL1910608)copy SMILEScopy InChI
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of Aurora A using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence micropl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355550(CHEMBL1910608)copy SMILEScopy InChI
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of CHK2 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355553(CHEMBL1910607)copy SMILEScopy InChI
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of Aurora A using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence micropl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355558(CHEMBL1910626)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355559(CHEMBL1910627)copy SMILEScopy InChI
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355560(CHEMBL1910628)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355561(CHEMBL1910629)copy SMILEScopy InChI
Affinity DataIC50: 3.13E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355562(CHEMBL1910630)copy SMILEScopy InChI
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355563(CHEMBL1910631)copy SMILEScopy InChI
Affinity DataIC50: 3.76E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355583(CHEMBL1910374)copy SMILEScopy InChI
Affinity DataIC50: 3.93E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355564(CHEMBL1910632)copy SMILEScopy InChI
Affinity DataIC50: 4.53E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355565(CHEMBL1910633)copy SMILEScopy InChI
Affinity DataIC50: 5.66E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355566(CHEMBL1910634)copy SMILEScopy InChI
Affinity DataIC50: 5.85E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355567(CHEMBL1910635)copy SMILEScopy InChI
Affinity DataIC50: 5.93E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355568(CHEMBL1910636)copy SMILEScopy InChI
Affinity DataIC50: 5.97E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355569(CHEMBL1910637)copy SMILEScopy InChI
Affinity DataIC50: 6.03E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355570(CHEMBL1910744)copy SMILEScopy InChI
Affinity DataIC50: 6.43E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355607(CHEMBL1910761)copy SMILEScopy InChI
Affinity DataIC50: 6.58E+3nMAssay Description:Inhibition of CHK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355571(CHEMBL1910745)copy SMILEScopy InChI
Affinity DataIC50: 7.32E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355556(CHEMBL1910623)copy SMILEScopy InChI
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Universit£ di Bologna

Curated by ChEMBL
LigandPNGBDBM50355551(CHEMBL1910371)copy SMILEScopy InChI
Affinity DataIC50: 8.26E+3nMAssay Description:Inhibition of RSK2 assessed as inhibition of substrate phosphorylation using fluorescent peptide substrate by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4R1DPubMed
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