Compile Data Set for Download or QSAR
Found 419 with Last Name = 'jane' and Initial = 'de'
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060627((S)-2-Amino-3-(5-iodo-2,4-dioxo-3,4-dihydro-2H-pyr...)copy SMILEScopy InChI
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060630((S)-2-Amino-3-(6-bromo-3,5-dioxo-4,5-dihydro-3H-[1...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060628((S)-2-Amino-3-(6-chloro-3,5-dioxo-4,5-dihydro-3H-[...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50111396(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2G89PubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060628((S)-2-Amino-3-(6-chloro-3,5-dioxo-4,5-dihydro-3H-[...)copy SMILEScopy InChI
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060630((S)-2-Amino-3-(6-bromo-3,5-dioxo-4,5-dihydro-3H-[1...)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060636((S)-2-Amino-3-(5-bromo-2,4-dioxo-3,4-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50111396(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)copy SMILEScopy InChI
Affinity DataKi:  11.6nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2G89PubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060628((S)-2-Amino-3-(6-chloro-3,5-dioxo-4,5-dihydro-3H-[...)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060630((S)-2-Amino-3-(6-bromo-3,5-dioxo-4,5-dihydro-3H-[1...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060629((S)-2-Amino-3-(6-iodo-3,5-dioxo-4,5-dihydro-3H-[1,...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060629((S)-2-Amino-3-(6-iodo-3,5-dioxo-4,5-dihydro-3H-[1,...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060630((S)-2-Amino-3-(6-bromo-3,5-dioxo-4,5-dihydro-3H-[1...)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060628((S)-2-Amino-3-(6-chloro-3,5-dioxo-4,5-dihydro-3H-[...)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50050704((R)-4-(3-Phosphono-propyl)-piperazine-2-carboxylic...)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060632((S)-2-Amino-3-(5-chloro-2,4-dioxo-3,4-dihydro-2H-p...)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060632((S)-2-Amino-3-(5-chloro-2,4-dioxo-3,4-dihydro-2H-p...)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060632((S)-2-Amino-3-(5-chloro-2,4-dioxo-3,4-dihydro-2H-p...)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50111396(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)copy SMILEScopy InChI
Affinity DataKi:  67nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2G89PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50419775(CHEMBL1950808)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060629((S)-2-Amino-3-(6-iodo-3,5-dioxo-4,5-dihydro-3H-[1,...)copy SMILEScopy InChI
Affinity DataKi:  74nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060633((S)-2-Amino-3-(6-methyl-3,5-dioxo-4,5-dihydro-3H-[...)copy SMILEScopy InChI
Affinity DataKi:  89nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060636((S)-2-Amino-3-(5-bromo-2,4-dioxo-3,4-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataKi:  92nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164540((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)copy SMILEScopy InChI
Affinity DataKi:  96nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2G89PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)copy SMILEScopy InChI
Affinity DataKi:  99.4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2G89PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9XTJPubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060636((S)-2-Amino-3-(5-bromo-2,4-dioxo-3,4-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataKi:  101nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060629((S)-2-Amino-3-(6-iodo-3,5-dioxo-4,5-dihydro-3H-[1,...)copy SMILEScopy InChI
Affinity DataKi:  101nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  103nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  107nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060631((S)-2-Amino-3-(5-nitro-2,4-dioxo-3,4-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataKi:  115nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  155nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060634((S)-2-Amino-3-(3,5-dioxo-4,5-dihydro-3H-[1,2,4]tri...)copy SMILEScopy InChI
Affinity DataKi:  163nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060627((S)-2-Amino-3-(5-iodo-2,4-dioxo-3,4-dihydro-2H-pyr...)copy SMILEScopy InChI
Affinity DataKi:  163nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060627((S)-2-Amino-3-(5-iodo-2,4-dioxo-3,4-dihydro-2H-pyr...)copy SMILEScopy InChI
Affinity DataKi:  176nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50002369((2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methyleth...)copy SMILEScopy InChI
Affinity DataKi:  177nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060634((S)-2-Amino-3-(3,5-dioxo-4,5-dihydro-3H-[1,2,4]tri...)copy SMILEScopy InChI
Affinity DataKi:  189nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060631((S)-2-Amino-3-(5-nitro-2,4-dioxo-3,4-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataKi:  207nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419775(CHEMBL1950808)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419775(CHEMBL1950808)copy SMILEScopy InChI
Affinity DataKi:  220nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2B receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060633((S)-2-Amino-3-(6-methyl-3,5-dioxo-4,5-dihydro-3H-[...)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2B receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9XTJPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2G89PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50050704((R)-4-(3-Phosphono-propyl)-piperazine-2-carboxylic...)copy SMILEScopy InChI
Affinity DataKi:  270nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Homo sapiens (Human))
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50060631((S)-2-Amino-3-(5-nitro-2,4-dioxo-3,4-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataKi:  279nMAssay Description:Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8MCBPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50004897((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)copy SMILEScopy InChI
Affinity DataKi:  280nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164555((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9XTJPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164555((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2G89PubMed
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