Compile Data Set for Download or QSAR
Found 208 with Last Name = 'böhmer' and Initial = 'fd'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359993(CHEMBL1928291)copy SMILEScopy InChI
Affinity DataIC50: 5.54nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359997(CHEMBL1928312)copy SMILEScopy InChI
Affinity DataIC50: 5.93nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359998(CHEMBL1928315)copy SMILEScopy InChI
Affinity DataIC50: 10.8nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359999(CHEMBL1928309)copy SMILEScopy InChI
Affinity DataIC50: 16.6nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359995(CHEMBL1928301)copy SMILEScopy InChI
Affinity DataIC50: 18.5nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359994(CHEMBL1928293)copy SMILEScopy InChI
Affinity DataIC50: 18.7nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359992(CHEMBL1928311)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of human FLT3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of endogenous FLT3 in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359996(CHEMBL1928310)copy SMILEScopy InChI
Affinity DataIC50: 43.7nMAssay Description:Inhibition of EGFR using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187340((6-Chloro-1H-indol-2-yl)-(5-methoxy-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of human PDGFR betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187345((5-Hydroxy-1H-indol-2-yl)-(4-methyl-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of endogenous FLT3 in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of Erbb2 using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187345((5-Hydroxy-1H-indol-2-yl)-(4-methyl-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of human FLT3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359992(CHEMBL1928311)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of EGFR autophosphorylation in EGF-stimulated human A431 cells after 1 hr by immunoblottingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antiproliferative activity against mouse 32Dcl3 cell line expressing wildtype FLT3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antiproliferative activity against mouse 32Dcl3 cell line expressing FLT3-ITDMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187369((5-Fluoro-1H-indol-2-yl)-(5-hydroxy-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of endogenous FLT3 in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 171nMAssay Description:Inhibition of human PDGFR betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM6581((5-Hydroxy-1H-2-indolyl)(1H-2-indolyl)-methanone |...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187340((6-Chloro-1H-indol-2-yl)-(5-methoxy-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50202219(5-hydroxybenzo[b]furan-2-yl-(5-hydroxy-1Hindol-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of endogenous PDGFRbeta autophosphorylation in Swiss 3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47NT9PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187357((4-Methyl-1H-indol-2-yl)-[5-(2-piperidin-1-yl-etho...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of human FLT3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50202219(5-hydroxybenzo[b]furan-2-yl-(5-hydroxy-1Hindol-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of endogenous FLT3 autophosphorylation in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47NT9PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50359999(CHEMBL1928309)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of EGFR autophosphorylation in EGF-stimulated human A431 cells after 1 hr by immunoblottingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of Erbb2 using poly(Glu,Tyr)4:1 as substrate and [gamma33P]ATP after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J966SRPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM6574((6-Methoxy-1H-2-indolyl)(1H-2-indolyl)methanone | ...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM6573((5-Methoxy-1H-2-indolyl)(1H-2-indolyl)methanone | ...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187365((4-Fluoro-1H-indol-2-yl)-(5-hydroxy-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of endogenous FLT3 in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetTubulin beta-2B chain(Bos taurus)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107672((3-Fluoro-phenyl)-(5-methoxy-1H-indol-2-yl)-methan...)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BZ65CNPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50202215((benzo[b]furan-2-yl)-(1H-indol-2-yl)methanone | CH...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of endogenous FLT3 autophosphorylation in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47NT9PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187348((5-Fluoro-1H-indol-2-yl)-(5-methoxy-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187345((5-Hydroxy-1H-indol-2-yl)-(4-methyl-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 458nMAssay Description:Inhibition of human PDGFR betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187345((5-Hydroxy-1H-indol-2-yl)-(4-methyl-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DNA synthesis in IL3 dependent FDC-P1 cells expressing wildtype KITMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DNA synthesis in IL3 dependent FDC-P1 cells expressing wildtype KITMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187345((5-Hydroxy-1H-indol-2-yl)-(4-methyl-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DNA synthesis in IL3 dependent FDC-P1 cells expressing KIT V558D mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187361((4-Chloro-1H-indol-2-yl)-(5-hydroxy-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187356((5-Fluoro-1H-indol-2-yl)-[5-(2-piperidin-1-yl-etho...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187351(Bis-(5-hydroxy-1H-indol-2-yl)-methanone | CHEMBL37...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DNA synthesis in IL3 dependent FDC-P1 cells expressing KIT V558D mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187366((5-Methoxy-1H-indol-2-yl)-(6-methyl-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetTubulin beta-2B chain(Bos taurus)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107658((5-Methoxy-1H-indol-2-yl)-phenyl-methanone | (5-me...)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107678((5-Methoxy-1H-indol-2-yl)-(3-methoxy-phenyl)-metha...)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BZ65CNPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187344((5-Hydroxy-1H-indol-2-yl)-(6-methoxy-1H-indol-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of endogenous FLT3 in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM6581((5-Hydroxy-1H-2-indolyl)(1H-2-indolyl)-methanone |...)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of endogenous FLT3 in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187367((5-Hydroxy-1H-indol-2-yl)-(6-methyl-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50187364((6-Fluoro-1H-indol-2-yl)-(5-hydroxy-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 590nMAssay Description:Inhibition of endogenous PDGFR in Swiss3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0M7BPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50202220(CHEMBL376787 | bis(5-aminobenzo[b]furan-2-yl)metha...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of endogenous FLT3 autophosphorylation in EOL1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47NT9PubMed
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