Compile Data Set for Download or QSAR
Found 58 with Last Name = 'bergé' and Initial = 'g'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19331(CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nM EC50:  3nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19333(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nM EC50:  0.600nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19332(N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nM EC50:  1.60nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19334(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-(2-ph...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nM EC50:  6.10nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19312((2S)-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nM Kd:  11nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19294(2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...)copy SMILEScopy InChI
Affinity DataIC50: 6nM Kd:  4nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19349(N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...)copy SMILEScopy InChI
Affinity DataIC50: 6nM Kd:  51nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19318(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1...)copy SMILEScopy InChI
Affinity DataIC50: 6.5nM EC50:  5.30nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19323((3R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 7nM EC50:  36nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19308((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataIC50: 9nM Kd:  6nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19310((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 9.5nM Kd:  13nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19321((3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataIC50: 10nM EC50:  2.5nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19326((2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 11nM Kd:  27nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19319(N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-...)copy SMILEScopy InChI
Affinity DataIC50: 13nM EC50:  9.90nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19293((R)-N-(1-(5-(2-(1H-Indol-3-yl)ethyl)-4-benzyl-4H-1...)copy SMILEScopy InChI
Affinity DataIC50: 15nM EC50:  64nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19322((3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 16nM Kd:  10nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19350(N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...)copy SMILEScopy InChI
Affinity DataIC50: 18nM EC50:  390nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19344(N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)e...)copy SMILEScopy InChI
Affinity DataIC50: 18nM EC50:  8.70nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19339(N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phenylet...)copy SMILEScopy InChI
Affinity DataIC50: 19nM EC50:  7.70nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19328((2R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 23nM Kd:  53nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19335(N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-...)copy SMILEScopy InChI
Affinity DataIC50: 24nM EC50:  5.40nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19309((2R)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataIC50: 28nM Kd:  7nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19327((2R)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataIC50: 29nM Kd:  8nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19296(2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 32nM Kd:  19nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19346((R,S)-N-((R)-1-(5-(2-(1H-Indol-3-yl)ethyl)-4-(2,4-...)copy SMILEScopy InChI
Affinity DataIC50: 32nM Kd:  5nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19311((2R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 32nM Kd:  8nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19347(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-(2-ph...)copy SMILEScopy InChI
Affinity DataIC50: 35nM EC50:  19.6nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19297(2-amino-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]...)copy SMILEScopy InChI
Affinity DataIC50: 38nM Kd:  27nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19313((2S)-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-...)copy SMILEScopy InChI
Affinity DataIC50: 44nM Kd:  32nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19325(N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1...)copy SMILEScopy InChI
Affinity DataIC50: 53nM Kd:  18nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19345(N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)m...)copy SMILEScopy InChI
Affinity DataIC50: 54nM EC50:  12nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19306((R)-N-(1-(4-(4-Methoxybenzyl)-5-phenethyl-4H-1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 59nM EC50:  256nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19340(N-[(1R)-1-[4-(2,4-dimethoxyphenyl)-5-(2-phenylethy...)copy SMILEScopy InChI
Affinity DataIC50: 63nM EC50:  14nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19337(N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)e...)copy SMILEScopy InChI
Affinity DataIC50: 70nM EC50:  2.30nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19338(N-[(1R)-1-[4-(4-ethylphenyl)-5-[2-(1H-indol-3-yl)e...)copy SMILEScopy InChI
Affinity DataIC50: 96nM EC50:  15nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19304((2S)-2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 113nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19324((3S)-N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phe...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19329((2R)-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-...)copy SMILEScopy InChI
Affinity DataIC50: 134nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19295(2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...)copy SMILEScopy InChI
Affinity DataIC50: 138nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19298(2-amino-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]...)copy SMILEScopy InChI
Affinity DataIC50: 154nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19317((2S,4R)-4-hydroxy-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[...)copy SMILEScopy InChI
Affinity DataIC50: 173nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19307((2S)-2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 175nM Kd:  24nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19348(N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phenylet...)copy SMILEScopy InChI
Affinity DataIC50: 178nM EC50:  143nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19303((2-aminoethyl)[(1R)-1-{4-[(2,4-dimethoxyphenyl)met...)copy SMILEScopy InChI
Affinity DataIC50: 190nM EC50:  279nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19342(N-[(1R)-2-(1H-indol-3-yl)-1-[5-(2-phenylethyl)-4-(...)copy SMILEScopy InChI
Affinity DataIC50: 255nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19305((2S)-2-amino-N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-...)copy SMILEScopy InChI
Affinity DataIC50: 275nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19316((2S)-N-[(1R)-1-[4-(4-ethylphenyl)-5-[2-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataIC50: 350nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19330((2R)-N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phe...)copy SMILEScopy InChI
Affinity DataIC50: 375nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19336(N-[(1R)-2-(1H-indol-3-yl)-1-[4-phenyl-5-(2-phenyle...)copy SMILEScopy InChI
Affinity DataIC50: 468nMAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
CNRS

LigandPNGBDBM19314((2S)-N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phe...)copy SMILEScopy InChI
Affinity DataIC50: 490nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7SZ4PubMed
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