Compile Data Set for Download or QSAR
Found 76 with Last Name = 'sagratini' and Initial = 'g'
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274054(CHEMBL4128084)copy SMILEScopy InChI
Affinity DataKi:  0.0398nMAssay Description:Displacement of [3H]prazosin from human alpha1D adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)copy SMILEScopy InChI
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMedDrugBank
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274049(CHEMBL342062)copy SMILEScopy InChI
Affinity DataKi:  0.0603nMAssay Description:Displacement of [3H]prazosin from human alpha1D adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274053(CHEMBL4126860)copy SMILEScopy InChI
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]prazosin from human alpha1D adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274049(CHEMBL342062)copy SMILEScopy InChI
Affinity DataKi:  0.0708nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMedDrugBank
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274053(CHEMBL4126860)copy SMILEScopy InChI
Affinity DataKi:  0.129nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50403649(CYCLAZOSIN)copy SMILEScopy InChI
Affinity DataKi:  0.135nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274061(CHEMBL4129461)copy SMILEScopy InChI
Affinity DataKi:  0.151nMAssay Description:Displacement of [3H]prazosin from human alpha1D adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274057(CHEMBL4129291)copy SMILEScopy InChI
Affinity DataKi:  0.151nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50403649(CYCLAZOSIN)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414396(CHEMBL564481)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274054(CHEMBL4128084)copy SMILEScopy InChI
Affinity DataKi:  0.191nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417541(CHEMBL1630938)copy SMILEScopy InChI
Affinity DataKi:  0.245nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274052(CHEMBL4127483)copy SMILEScopy InChI
Affinity DataKi:  0.302nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50403649(CYCLAZOSIN)copy SMILEScopy InChI
Affinity DataKi:  0.324nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417542(CHEMBL1630939)copy SMILEScopy InChI
Affinity DataKi:  0.324nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417541(CHEMBL1630938)copy SMILEScopy InChI
Affinity DataKi:  0.339nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417542(CHEMBL1630939)copy SMILEScopy InChI
Affinity DataKi:  0.347nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274050(CHEMBL4125981)copy SMILEScopy InChI
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274057(CHEMBL4129291)copy SMILEScopy InChI
Affinity DataKi:  0.389nMAssay Description:Displacement of [3H]prazosin from human alpha1D adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414396(CHEMBL564481)copy SMILEScopy InChI
Affinity DataKi:  0.417nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414397(CHEMBL558890)copy SMILEScopy InChI
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274054(CHEMBL4128084)copy SMILEScopy InChI
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM86731(CAS_74191-85-8 | Doxazosin | UK 33,274)copy SMILEScopy InChI
Affinity DataKi:  0.537nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMedDrugBank
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274049(CHEMBL342062)copy SMILEScopy InChI
Affinity DataKi:  0.589nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417540(CHEMBL1630940)copy SMILEScopy InChI
Affinity DataKi:  0.603nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)copy SMILEScopy InChI
Affinity DataKi:  0.631nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50403649(CYCLAZOSIN)copy SMILEScopy InChI
Affinity DataKi:  0.692nMAssay Description:Binding affinity to human alpha1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274061(CHEMBL4129461)copy SMILEScopy InChI
Affinity DataKi:  0.741nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274059(CHEMBL4128460)copy SMILEScopy InChI
Affinity DataKi:  0.776nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM86731(CAS_74191-85-8 | Doxazosin | UK 33,274)copy SMILEScopy InChI
Affinity DataKi:  0.813nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM86731(CAS_74191-85-8 | Doxazosin | UK 33,274)copy SMILEScopy InChI
Affinity DataKi:  0.813nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMedDrugBank
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274057(CHEMBL4129291)copy SMILEScopy InChI
Affinity DataKi:  0.871nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274060(CHEMBL4127078)copy SMILEScopy InChI
Affinity DataKi:  0.912nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414399(CHEMBL561851)copy SMILEScopy InChI
Affinity DataKi:  0.933nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417540(CHEMBL1630940)copy SMILEScopy InChI
Affinity DataKi:  0.955nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274055(CHEMBL4125846)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414396(CHEMBL564481)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Binding affinity to alpha1B adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414397(CHEMBL558890)copy SMILEScopy InChI
Affinity DataKi:  1.41nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414399(CHEMBL561851)copy SMILEScopy InChI
Affinity DataKi:  1.58nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414399(CHEMBL561851)copy SMILEScopy InChI
Affinity DataKi:  1.86nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274053(CHEMBL4126860)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417541(CHEMBL1630938)copy SMILEScopy InChI
Affinity DataKi:  1.91nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50417542(CHEMBL1630939)copy SMILEScopy InChI
Affinity DataKi:  2.09nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3GNTPubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50274055(CHEMBL4125846)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]prazosin from human alpha1D adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414396(CHEMBL564481)copy SMILEScopy InChI
Affinity DataKi:  2.82nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50403649(CYCLAZOSIN)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]prazosin from human alpha1D adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414397(CHEMBL558890)copy SMILEScopy InChI
Affinity DataKi:  3.39nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ88W5PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ di Camerino

Curated by ChEMBL
LigandPNGBDBM50414396(CHEMBL564481)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Binding affinity to alpha1A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92DS4PubMed
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