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Found 273 with Last Name = 'tanabe' and Initial = 'g'
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612995(CHEMBL5276586)copy SMILES
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612998(CHEMBL5269400)copy SMILES
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50613001(CHEMBL5268739)copy SMILES
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50613004(CHEMBL5282029)copy SMILES
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612994(CHEMBL5283777)copy SMILES
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612995(CHEMBL5276586)copy SMILES
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612998(CHEMBL5269400)copy SMILES
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50613001(CHEMBL5268739)copy SMILES
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50613004(CHEMBL5282029)copy SMILES
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612994(CHEMBL5283777)copy SMILES
Affinity DataKi:  0.840nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147013(CHEMBL3764559)copy SMILEScopy InChI
Affinity DataKi:  185nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B92NFPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147016(CHEMBL3763300)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147107(CHEMBL3763319)copy SMILEScopy InChI
Affinity DataKi:  216nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147158(CHEMBL3764745)copy SMILEScopy InChI
Affinity DataKi:  353nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147159(CHEMBL3764813)copy SMILEScopy InChI
Affinity DataKi:  785nMAssay Description:Competitive inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50549692(CHEMBL4749306)copy SMILES
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B92NFPubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50549691(CHEMBL4754034)copy SMILES
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B92NFPubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50549693(CHEMBL4750690)copy SMILES
Affinity DataKi:  5.10E+4nMAssay Description:Inhibition of recombinant human maltase-glucoamylase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 35 mins by microtiter pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B92NFPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180584(CHEMBL3814496)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180582(CHEMBL3814988)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180583(CHEMBL3815109)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612995(CHEMBL5276586)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50342937((1S,2R,3S,4S)-1-((2S,3S)-3-ethoxy-2,4-dihydroxybut...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RJCPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180520(CHEMBL3814838)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50342939((1S,2R,3S,4S)-1-((2S,3S)-3-(benzyloxy)-2,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RJCPubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50180584(CHEMBL3814496)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1044CPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RJCPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)copy SMILEScopy InChI
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
In DepthDetails
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9J8RPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147107(CHEMBL3763319)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612995(CHEMBL5276586)copy SMILES
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147014(CHEMBL3764223)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180584(CHEMBL3814496)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612998(CHEMBL5269400)copy SMILES
Affinity DataIC50: 220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetLysosomal alpha-glucosidase(Rattus norvegicus)TBA
LigandPNGBDBM50612998(CHEMBL5269400)copy SMILES
Affinity DataIC50: 230nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180580(CHEMBL3814911)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180580(CHEMBL3814911)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50342937((1S,2R,3S,4S)-1-((2S,3S)-3-ethoxy-2,4-dihydroxybut...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RJCPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180520(CHEMBL3814838)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147012(CHEMBL3763591)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180583(CHEMBL3815109)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50327501(CHEMBL1258528 | ponkoranol)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1044CPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9J8RPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50180586(CHEMBL1182462)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q241700VPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50338676(1,4-Dideoxy-1,4-{(R)-[(2S,3R,4R,5S)-2,3,4,5,6-pent...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1044CPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of rat intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1044CPubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50612999(CHEMBL5277322)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50147008(CHEMBL3765363)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0WSHPubMed
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