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Found 98 with Last Name = 'kang' and Initial = 'je'
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50355214(CHEMBL401566)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50355210(CHEMBL1835715)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50355212(CHEMBL1835717)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50355211(CHEMBL1835716)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50355213(CHEMBL1835792)copy SMILEScopy InChI
Affinity DataKi:  1.35E+3nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50311585(CHEMBL455372 | Erythrabyssin II | erybraedin C)copy SMILEScopy InChI
Affinity DataKi:  2.73E+3nMAssay Description:Non-competitive inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by Linewe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405744(CHEMBL5274088)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405742(CHEMBL5271520)copy SMILEScopy InChI
Affinity DataIC50: 6.40nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) obtained from human WIL2 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405753(CHEMBL5274634)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405753(CHEMBL5274634)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405681(CHEMBL5271793)copy SMILEScopy InChI
Affinity DataIC50: 8.70nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405679(CHEMBL5266236)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405680(CHEMBL5268616)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405750(CHEMBL5291256)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405746(CHEMBL5286013)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) obtained from human WIL2 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405748(CHEMBL5279952)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50380399(CHEMBL2018302 | Tubastatin A | US10227295, Compoun...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50380399(CHEMBL2018302 | Tubastatin A | US10227295, Compoun...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405757(CHEMBL5271343)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405751(CHEMBL5281142)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405747(CHEMBL5267739)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405739(CHEMBL5273396)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405745(CHEMBL5285879)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405740(CHEMBL5280669)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) obtained from human WIL2 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405743(CHEMBL5274632)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405756(CHEMBL5284689)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405758(CHEMBL5287109)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405741(CHEMBL5271970)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against thymidylate synthase isolated from L1210 leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405752(CHEMBL5290601)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405749(CHEMBL5285996)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405678(CHEMBL5287254)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) obtained from human WIL2 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails DrugBank
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails DrugBank
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50355214(CHEMBL401566)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405677(CHEMBL5267379)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) obtained from human WIL2 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405742(CHEMBL5271520)copy SMILEScopy InChI
Affinity DataIC50: 111nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405744(CHEMBL5274088)copy SMILEScopy InChI
Affinity DataIC50: 122nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 132nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 132nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405748(CHEMBL5279952)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50405755(CHEMBL5281671)copy SMILEScopy InChI
Affinity DataIC50: 152nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 2(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 164nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405746(CHEMBL5286013)copy SMILEScopy InChI
Affinity DataIC50: 167nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405743(CHEMBL5274632)copy SMILEScopy InChI
Affinity DataIC50: 168nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetSialidase(Clostridium perfringens)
Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50355212(CHEMBL1835717)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of Clostridium perfringens neuraminidase using 4-methylumbelliferyl-alpha-D-N-acetylneuraminic acid as substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53M8XPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405747(CHEMBL5267739)copy SMILEScopy InChI
Affinity DataIC50: 197nMAssay Description:Inhibitory activity against acetylcholinetransferase (AChE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405679(CHEMBL5266236)copy SMILEScopy InChI
Affinity DataIC50: 206nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50405745(CHEMBL5285879)copy SMILEScopy InChI
Affinity DataIC50: 212nMAssay Description:Inhibition of choline acetyltransferase (CAT) enzymeMore data for this Ligand-Target Pair
In DepthDetails
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