Compile Data Set for Download or QSAR
Found 310 with Last Name = 'mack' and Initial = 'jf'
TargetHexokinase-2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50169013(CHEMBL3805703)copy SMILEScopy InChI
Affinity DataKi:  2.90E+3nMAssay Description:Competitive inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) assessed as formation of G6P by continuou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XWWPubMed
LigandPNGBDBM50420316(CHEMBL2089119)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420311(CHEMBL2089114)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420321(CHEMBL2089112)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420309(CHEMBL2089120)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420317(CHEMBL2089118)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420310(CHEMBL2089116)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420312(CHEMBL2089109)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420313(CHEMBL2089108)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420314(CHEMBL2089107)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420315(CHEMBL2089106)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365868(CHEMBL1957857)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365882(CHEMBL1957870)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420311(CHEMBL2089114)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420316(CHEMBL2089119)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365867(CHEMBL1957856)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365869(CHEMBL1957858)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420309(CHEMBL2089120)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365865(CHEMBL1957841)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420321(CHEMBL2089112)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365866(CHEMBL1957855)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420324(CHEMBL2089105)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420325(CHEMBL2089104)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420322(CHEMBL2089111)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420320(CHEMBL2089113)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365882(CHEMBL1957870)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3Kdelta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365873(CHEMBL1957862)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420318(CHEMBL2089117)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365880(CHEMBL1957868)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365890(CHEMBL1957875)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3KbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365872(CHEMBL1957861)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
TargetHexokinase-1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50169033(CHEMBL3806069)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XWWPubMed
TargetHexokinase-1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50169038(CHEMBL3804841)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XWWPubMed
TargetHexokinase-2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50169042(CHEMBL3806103)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XWWPubMed
LigandPNGBDBM50420319(CHEMBL2089115)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365870(CHEMBL1957859)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365868(CHEMBL1957857)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of PI3Kdelta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420314(CHEMBL2089107)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420310(CHEMBL2089116)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420317(CHEMBL2089118)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
TargetHexokinase-2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50169037(CHEMBL3805205)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XWWPubMed
LigandPNGBDBM50420326(CHEMBL2089103)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365884(CHEMBL1957872)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365880(CHEMBL1957868)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kdelta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420313(CHEMBL2089108)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365864(CHEMBL1957840)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365871(CHEMBL1957860)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365878(CHEMBL1957866)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365878(CHEMBL1957866)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365878(CHEMBL1957866)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of PI3Kdelta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
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