Compile Data Set for Download or QSAR
Found 117 with Last Name = 'kikuchi' and Initial = 'k'
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)copy SMILEScopy InChI
Affinity DataKi:  8.30nMAssay Description:Antagonist activity at human CRF1 receptor expressed in IMR32 cells assessed as inhibition of CRF-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420920(CHEMBL2087549 | CHEMBL2087567)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Antagonist activity at human CRF1 receptor expressed in IMR32 cells assessed as inhibition of CRF-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420920(CHEMBL2087549 | CHEMBL2087567)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human CRF2 receptor expressed in IMR32 cells assessed as inhibition of CRF-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50084833(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:Binding affinity for Retinoic Acid Receptor alpha (RAR alpha)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]-ATRA-Hl60 binding to Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23T9GFVPubMedMMDB
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Binding affinity against Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028QSBPubMedMMDB
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.780nMAssay Description:Inhibition of [3H]-ATRA-Hl60 binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23T9GFVPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.890nMAssay Description:Binding affinity for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028QSBPubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of [3H]-ATRA-Hl60 binding to Retinoic acid receptor betaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23T9GFVPubMedMMDB
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.940nMAssay Description:Binding affinity for Retinoic acid receptor betaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028QSBPubMedMMDB
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084832(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50084835(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Binding affinity for Retinoic Acid Receptor alpha (RAR alpha)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50084832(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Binding affinity for Retinoic Acid Receptor alpha (RAR alpha)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084834(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084830(4-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084832(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084831(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420904(CHEMBL2087550)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420906(CHEMBL2087552)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420908(CHEMBL2087554)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420909(CHEMBL2087555)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420905(CHEMBL2087551)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084829(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50084834(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Binding affinity for Retinoic Acid Receptor alpha (RAR alpha)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420912(CHEMBL2087558)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420916(CHEMBL2087562)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human CRF1 receptor expressed in HEK293 cells assessed as inhibition of CRF-stimulated cAMP accumulation after 30 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084830(4-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084833(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420916(CHEMBL2087562)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420915(CHEMBL2087561)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420920(CHEMBL2087549 | CHEMBL2087567)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human CRF1 receptor expressed in HEK293 cells assessed as inhibition of CRF-stimulated cAMP accumulation after 30 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420907(CHEMBL2087553)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420930(CHEMBL2087795)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420935(CHEMBL2087799)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084834(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420927(CHEMBL2087574)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human CRF1 receptor expressed in HEK293 cells assessed as inhibition of CRF-stimulated cAMP accumulation after 30 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50099474(4-[5-(8-Isopropyl-4-phenyl-quinolin-2-yl)-1H-pyrro...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Antagonistic activity of the compound was evaluated in terms of inhibition of Retinoic acid receptor alpha transactivation by ATRA (50 nM)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M3643PubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50084831(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Binding affinity for Retinoic Acid Receptor alpha (RAR alpha)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420914(CHEMBL2087560)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420937(CHEMBL2087801)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420927(CHEMBL2087574)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084829(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420913(CHEMBL2087559)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420931(CHEMBL2087796)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human CRF1 receptor expressed in HEK293 cells assessed as inhibition of CRF-stimulated cAMP accumulation after 30 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084831(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Binding affinity for Retinoic Acid Receptor beta (RAR beta)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420917(CHEMBL2087563)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50084836(4-[(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quinoxa...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Binding affinity for Retinoic Acid Receptor alpha (RAR alpha).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420924(CHEMBL2087571)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50420911(CHEMBL2087557)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32XCPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Binding affinity for Retinoic Acid Receptor alpha (RAR alpha)More data for this Ligand-Target Pair
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