BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor alpha' and Ligand = 'BDBM50099474'

Retinoic acid receptor alpha(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL

BDBM50099474(4-[5-(8-Isopropyl-4-phenyl-quinolin-2-yl)-1H-pyrro...)copy SMILEScopy InChI

IC50: 31nMAssay Description:Antagonistic activity of the compound was evaluated in terms of inhibition of Retinoic acid receptor alpha transactivation by ATRA (50 nM)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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B.MOAD DrugBank antibodypedia GoogleScholar

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Details
BindingDB Entry DOI: 10.7270/Q26M3643PubMed