Compile Data Set for Download or QSAR
Found 209 with Last Name = 'stebbins' and Initial = 'kj'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M1 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M3 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M4 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  19nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M2 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataIC50: 1.58nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50366775(BENZTROPINE | Benzatropine)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M4 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549908(CHEMBL4760610)copy SMILES
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549901(CHEMBL4799006)copy SMILES
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549929(CHEMBL4755122)copy SMILES
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549893(CHEMBL4757103)copy SMILES
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549908(CHEMBL4760610)copy SMILES
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549901(CHEMBL4799006)copy SMILES
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549929(CHEMBL4755122)copy SMILES
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549896(CHEMBL4784357)copy SMILES
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549896(CHEMBL4784357)copy SMILES
Affinity DataIC50: 8.70nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549898(CHEMBL4799613)copy SMILES
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549898(CHEMBL4799613)copy SMILES
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549892(CHEMBL4742997)copy SMILES
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549892(CHEMBL4742997)copy SMILES
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508126(CHEMBL4457564)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508159(CHEMBL4529735)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508153(CHEMBL4549922)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508137(CHEMBL4437146)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549903(CHEMBL4779636)copy SMILES
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549926(CHEMBL4783670)copy SMILES
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))TBA
LigandPNGBDBM50366775(BENZTROPINE | Benzatropine)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M3 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549903(CHEMBL4779636)copy SMILES
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M4 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549902(CHEMBL4755240)copy SMILES
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549926(CHEMBL4783670)copy SMILES
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508144(CHEMBL4545223)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549902(CHEMBL4755240)copy SMILES
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M4 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508159(CHEMBL4529735)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549919(CHEMBL4797503)copy SMILES
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549939(CHEMBL4788792)copy SMILES
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549919(CHEMBL4797503)copy SMILES
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508127(CHEMBL4449687)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508145(CHEMBL4450146)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549895(CHEMBL4747295)copy SMILES
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549894(CHEMBL4743811)copy SMILES
Affinity DataIC50: 31.6nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549907(CHEMBL4794536)copy SMILES
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549907(CHEMBL4794536)copy SMILES
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549894(CHEMBL4743811)copy SMILES
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549895(CHEMBL4747295)copy SMILES
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508147(CHEMBL4530053)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508151(CHEMBL4449183)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508126(CHEMBL4457564)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549924(CHEMBL4763789)copy SMILES
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
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