Compile Data Set for Download or QSAR
Found 35 with Last Name = 'cleghorn' and Initial = 'la'
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364113(CHEMBL1230468)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Leishmania major N-myristoyltransferase using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364113(CHEMBL1230468)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364135(CHEMBL1951295)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364127(CHEMBL1951287)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50384600(CHEMBL2036792 | US9744172, Compound UNC00000563A)copy SMILEScopy InChI
Affinity DataIC50: 114nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364136(CHEMBL1951296)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50384600(CHEMBL2036792 | US9744172, Compound UNC00000563A)copy SMILEScopy InChI
Affinity DataIC50: 199nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364133(CHEMBL1951293)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364121(CHEMBL1951280)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364122(CHEMBL1951282)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364123(CHEMBL1951283)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364126(CHEMBL1951286)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364124(CHEMBL1951284)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364117(CHEMBL1951274)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364131(CHEMBL1951291)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364134(CHEMBL1951294)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50517286(CHEMBL4516798)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 20 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364118(CHEMBL1951277)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364125(CHEMBL1951285)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364129(CHEMBL1951289)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364128(CHEMBL1951288)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364119(CHEMBL1951278)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364116(CHEMBL1951273)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50517286(CHEMBL4516798)copy SMILEScopy InChI
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50517285(CHEMBL4572962)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CDK4 by kinobeads-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364114(CHEMBL1951105)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364113(CHEMBL1230468)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human ERG by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50517285(CHEMBL4572962)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50517287(CHEMBL4563818)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50517285(CHEMBL4572962)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 20 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50517287(CHEMBL4563818)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 20 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC867RPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364132(CHEMBL1951292)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364120(CHEMBL1951279)copy SMILEScopy InChI
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364115(CHEMBL1951272)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50364130(CHEMBL1951290)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed