Compile Data Set for Download or QSAR
Found 12 with Last Name = 'jr.' and Initial = 'lj'
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423465(US11753373, Compound A-1-c | WO2006061714, P38.8 |...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nM EC50:  4.20E+6nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423464(WO2006061714, P38.7 | WO2006061714-ID-09 | cmdc.20...)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+4nM EC50:  3.60E+6nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423469(WO2006061714, P39.4 | WO2006061714-ID-14 | cmdc.20...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nM EC50:  1.80E+7nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423466(WO2006061714, P39.1 | WO2006061714-ID-11 | cmdc.20...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+4nM EC50:  2.50E+7nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM442803(WO2006061714, P38.5 | cmdc.202100576, 10f)copy SMILES
Affinity DataIC50: 2.30E+6nM EC50:  9.15E+7nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423467(WO2006061714, P39.2 | WO2006061714-ID-12)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+7nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423468(WO2006061714, P39.3 | WO2006061714-ID-13)copy SMILEScopy InChI
Affinity DataIC50: 9.70E+7nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423470(WO2006061714, P39.5 | WO2006061714-ID-15)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+8nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423460(WO2006061714, Example 2 | WO2006061714-ID-02)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+8nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423462(US11753373, Compound A-5-a | WO2006061714, P38.2 |...)copy SMILEScopy InChI
Affinity DataEC50:  1.40E+6nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM442796(WO2006061714, P38.1)copy SMILES
Affinity DataEC50:  8.00E+5nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed
TargetReplicase polyprotein 1ab(SARS coronavirus Urbani)
Pfizer Inc.

LigandPNGBDBM423459(WO2006061714, Example 1 | WO2006061714-ID-01)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+8nMAssay Description:Proteolytic activity of Coronavirus 3C protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS 3CI_pro FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2K5WPubMed