TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]DTG from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Inhibition of BBOX (unknown origin)More data for this Ligand-Target Pair
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 0.0500nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Binding affinity to human neuropeptide Y1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Binding affinity to human neuropeptide Y2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Binding affinity to NTS1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Binding affinity to human NK1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Binding affinity to ORL1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Binding affinity to human histamine H1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to human dopamine D2S receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity to human glucocorticoid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity to human NK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Binding affinity to human 5-HT3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Binding affinity to human NK3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity to human bradykinin B2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity to PGI2 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute of Organic Synthesis
Curated by ChEMBL
Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Displacement of [3H]1,3-di(2-tolyl)guanidine from sigma 1 receptor in human Jurkat cellsMore data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Binding affinity to human histamine H2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.17E+5nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Latvian Biomedical Research and Study centre
Curated by ChEMBL
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair