Compile Data Set for Download or QSAR
Found 48 with Last Name = 'gozelle' and Initial = 'm'
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50247128((6,6-dimethyl-5,6-dihydroimidazo[2,1-b][1,3]thiazo...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50247128((6,6-dimethyl-5,6-dihydroimidazo[2,1-b][1,3]thiazo...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of CXCL12-red from human NLuc-tagged CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50247128((6,6-dimethyl-5,6-dihydroimidazo[2,1-b][1,3]thiazo...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human DEF3-RLuc fused CXCR4 receptor expressed in HEK293T cells co-expressing DEF3-Beta-arrestin-2-mVenus assessed as inhibiti...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50247128((6,6-dimethyl-5,6-dihydroimidazo[2,1-b][1,3]thiazo...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human DEF3-fused CXCR4 receptor expressed in HEK293T cells co-expressing DAN1-HA-Galphaq/i5 assessed as inhibition of CXCL12-i...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521156(CHEMBL4452433)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50035696(1,1''-{1,4-phenylenebis(methylene)}-bis{1,4,8,11-t...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521159(CHEMBL4533528)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521148(CHEMBL4444949)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521158(CHEMBL4463564)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521164(CHEMBL4558842)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521143(CHEMBL4557428)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521160(CHEMBL4585865)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521144(CHEMBL4514484)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521161(CHEMBL4438705)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521142(CHEMBL4438964)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521168(CHEMBL4445831)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521142(CHEMBL4438964)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Displacement of CXCL12-red from human NLuc-tagged CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521145(CHEMBL4548557)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521144(CHEMBL4514484)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Displacement of CXCL12-red from human NLuc-tagged CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521166(CHEMBL4539571)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521162(CHEMBL4440964)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521156(CHEMBL4452433)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human DEF3-fused CXCR4 receptor expressed in HEK293T cells co-expressing DAN1-HA-Galphaq/i5 assessed as inhibition of CXCL12-i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521165(CHEMBL4561387)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521149(CHEMBL4529593)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521156(CHEMBL4452433)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of CXCL12-red from human NLuc-tagged CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521142(CHEMBL4438964)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human DEF3-fused CXCR4 receptor expressed in HEK293T cells co-expressing DAN1-HA-Galphaq/i5 assessed as inhibition of CXCL12-i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521150(CHEMBL4463569)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521151(CHEMBL4526858)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521144(CHEMBL4514484)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human DEF3-fused CXCR4 receptor expressed in HEK293T cells co-expressing DAN1-HA-Galphaq/i5 assessed as inhibition of CXCL12-i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521152(CHEMBL4465129)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521147(CHEMBL4585203)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521171(CHEMBL4450496)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521142(CHEMBL4438964)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Antagonist activity at human DEF3-RLuc fused CXCR4 receptor expressed in HEK293T cells co-expressing DEF3-Beta-arrestin-2-mVenus assessed as inhibiti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521156(CHEMBL4452433)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human DEF3-RLuc fused CXCR4 receptor expressed in HEK293T cells co-expressing DEF3-Beta-arrestin-2-mVenus assessed as inhibiti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521170(CHEMBL4566356)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521144(CHEMBL4514484)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+3nMAssay Description:Antagonist activity at human DEF3-RLuc fused CXCR4 receptor expressed in HEK293T cells co-expressing DEF3-Beta-arrestin-2-mVenus assessed as inhibiti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521167(CHEMBL4536186)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521154(CHEMBL4443602)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521153(CHEMBL4463684)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521146(CHEMBL4460308)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521169(CHEMBL4469048)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521141(CHEMBL4454166)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521155(CHEMBL4461446)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521157(CHEMBL4531030)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521163(CHEMBL4469779)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50461977(CHEMBL4226649)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR4 receptor expressed in HEK293T cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521157(CHEMBL4531030)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Antagonist activity at human DEF3-fused CXCR4 receptor expressed in HEK293T cells co-expressing DAN1-HA-Galphaq/i5 assessed as inhibition of CXCL12-i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Griffin Discoveries BV

Curated by ChEMBL
LigandPNGBDBM50521157(CHEMBL4531030)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Antagonist activity at human DEF3-RLuc fused CXCR4 receptor expressed in HEK293T cells co-expressing DEF3-Beta-arrestin-2-mVenus assessed as inhibiti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72V6PubMed