Compile Data Set for Download or QSAR
Found 223 with Last Name = 'lanza' and Initial = 'm'
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50435130(CHEMBL1893324)copy SMILEScopy InChI
Affinity DataKi:  0.0670nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50015490(CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITR...)copy SMILEScopy InChI
Affinity DataKi:  0.0760nMAssay Description:Binding affinity to human neuropeptide Y receptor type 2 by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50015490(CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITR...)copy SMILEScopy InChI
Affinity DataKi:  0.0960nMAssay Description:Binding affinity to human neuropeptide Y receptor type 1 by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50335566(CHEMBL1651026 | Substance P [Sar9,Met(O2)11])copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human NK1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)copy SMILEScopy InChI
Affinity DataKi:  0.270nMAssay Description:Binding affinity to human NTS1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)copy SMILEScopy InChI
Affinity DataKi:  0.460nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50333104(CHEMBL389521 | H-FGGFTGARKSARKLANQ-NH2 | N/OFQ-NH2...)copy SMILEScopy InChI
Affinity DataKi:  0.480nMAssay Description:Binding affinity to human NOP receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50366495((+)butaclamol | CHEMBL1255588)copy SMILEScopy InChI
Affinity DataKi:  0.740nMAssay Description:Binding affinity to human dopamine D2S receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)copy SMILEScopy InChI
Affinity DataKi:  0.950nMAssay Description:Binding affinity to human histamine H1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMedDrugBank
TargetGlucocorticoid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human glucocorticoid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGalanin receptor type 2(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50051295((S)-3-methyl-2-phenyl-N-(1-phenylpropyl)quinoline-...)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human NK3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM82561(CAS_40796-97-2 | TROPANYL 3,5-DICHLOROBENZOATE | T...)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Binding affinity to human 5-HT3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM23954(5-[(2E,3aS,4R,5R,6aS)-5-hydroxy-4-[(1E,3S)-3-hydro...)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human PGI2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50435131(CHEMBL2390989)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Binding affinity to human NK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420342(CHEMBL2089156)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50435129(CHEMBL2392354)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Binding affinity to human bradykinin B2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493433(CHEMBL2431282)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419880(CHEMBL1956197)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50056415(2-piperidinopropyl 4-amino-5-chloro-2-methoxybenzo...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Displacement of [3H]GR113808 from Dunkin-Hartley guinea pig brain striatum 5HT4R after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z45ZQPubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50388686(CHEMBL74656)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]GR113808 from Dunkin-Hartley guinea pig brain striatum 5HT4R after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z45ZQPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50019529(CHEMBL3291085)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Binding affinity to 5HT4R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z45ZQPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420341(CHEMBL2089155)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420342(CHEMBL2089156)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50019523(CHEMBL3291078)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Displacement of [3H]GR113808 from Dunkin-Hartley guinea pig brain striatum 5HT4R after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z45ZQPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50420341(CHEMBL2089155)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417345(CHEMBL1276219)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473179(CHEMBL13917)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493433(CHEMBL2431282)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50019520(CHEMBL3291075)copy SMILEScopy InChI
Affinity DataKi:  52nMAssay Description:Displacement of [3H]GR113808 from Dunkin-Hartley guinea pig brain striatum 5HT4R after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z45ZQPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataKi:  52nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)copy SMILEScopy InChI
Affinity DataKi:  58nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473154(CHEMBL14107)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473154(CHEMBL14107)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493430(CHEMBL2431281)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50493431(CHEMBL2431280)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
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