Compile Data Set for Download or QSAR
Found 137 with Last Name = 'iwamura' and Initial = 'n'
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461646(CHEBI:582124 | Myriocin)copy SMILEScopy InChI
Affinity DataIC50: 0.130nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248627(CHEMBL4078454)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of full length recombinant human His-tagged CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248633(CHEMBL4083552)copy SMILEScopy InChI
Affinity DataIC50: 0.340nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461644(CHEMBL4228416)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248645(CHEMBL4061525)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248623(CHEMBL4096487)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of full length recombinant human His-tagged CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248614(CHEMBL4066819)copy SMILEScopy InChI
Affinity DataIC50: 0.460nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248635(CHEMBL4070408)copy SMILEScopy InChI
Affinity DataIC50: 0.470nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461649(CHEMBL4225519)copy SMILEScopy InChI
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248633(CHEMBL4083552)copy SMILEScopy InChI
Affinity DataIC50: 0.550nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248656(CHEMBL4086487)copy SMILEScopy InChI
Affinity DataIC50: 0.570nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248656(CHEMBL4086487)copy SMILEScopy InChI
Affinity DataIC50: 0.570nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248645(CHEMBL4061525)copy SMILEScopy InChI
Affinity DataIC50: 0.590nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248640(CHEMBL4074204)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248690(CHEMBL4082469)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461645(CHEMBL4228472)copy SMILEScopy InChI
Affinity DataIC50: 0.710nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248635(CHEMBL4070408)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248611(CHEMBL4060856)copy SMILEScopy InChI
Affinity DataIC50: 0.930nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248611(CHEMBL4060856)copy SMILEScopy InChI
Affinity DataIC50: 0.970nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248638(CHEMBL4062244)copy SMILEScopy InChI
Affinity DataIC50: 0.990nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248614(CHEMBL4066819)copy SMILEScopy InChI
Affinity DataIC50: 0.990nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248612(CHEMBL4076395)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248615(CHEMBL4077627)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248640(CHEMBL4074204)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461647(CHEMBL4225462)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461643(CHEMBL4225764)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248690(CHEMBL4082469)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248638(CHEMBL4062244)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248686(CHEMBL4071040)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248686(CHEMBL4071040)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248662(CHEMBL4091345)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248615(CHEMBL4077627)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248612(CHEMBL4076395)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248632(CHEMBL4069854)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248687(CHEMBL4090775)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248687(CHEMBL4090775)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248662(CHEMBL4091345)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248632(CHEMBL4069854)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248690(CHEMBL4082469)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248609(CHEMBL4088931)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248658(CHEMBL4060714)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461639(CHEMBL4229253)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461641(CHEMBL4225192)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248639(CHEMBL4072372)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248658(CHEMBL4060714)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248628(CHEMBL4072496)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of full length recombinant human His-tagged CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ...More data for this Ligand-Target Pair
TargetSerine palmitoyltransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50461638(CHEMBL4226297)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Inhibition of human SPT2 transfected in Freestyle293 cells using L-serine and palmitoyl-CoA as substrate preincubated for 60 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XNHPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248639(CHEMBL4072372)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248678(CHEMBL4062262)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50248609(CHEMBL4088931)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9D6HPubMed
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