Compile Data Set for Download or QSAR
Found 230 with Last Name = 'robinson' and Initial = 'pj'
TargetMelanocortin receptor 4(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50128358(CHEMBL3629347)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Inhibition of human recombinant melanocortin 4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)copy SMILEScopy InChI
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]4-DAMP from human recombinant Muscarinic acetylcholine receptor M3 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)copy SMILEScopy InChI
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]methyl-spiperone from human recombinant D2S receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)copy SMILEScopy InChI
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)copy SMILEScopy InChI
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]U 69593 from rat recombinant kappa opioid receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)copy SMILEScopy InChI
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMedDrugBank
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM28582(1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine | CHE...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I](+/-)DOI from human recombinant 5-HT2B receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetSubstance-K receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233962(CHEMBL4068783)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [125I]NKA from human recombinant tachykinin NK2 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50176062(3-(5H-dibenzo[a,d][7]annulen-5-yl)-N-methylpropan-...)copy SMILEScopy InChI
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]nisoxetine from human recombinant norepinephrine transporter expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMedDrugBank
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50005534(1-(1-(benzo[b]thiophen-2-yl)cyclohexyl)piperidine ...)copy SMILEScopy InChI
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]BTCP from human recombinant dopamine transporter expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Displacement of [3H]pirenzepine from human recombinant Muscarinic acetylcholine receptor M1 expressed in CHO cells after 60 mins by scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  61nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT5a receptor in HEK293 cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM181119(US9138393, Cimetidine | US9144538, Cimetidine)copy SMILEScopy InChI
Affinity DataKi:  490nMAssay Description:Displacement of [125I]APT from human recombinant histamine H2 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50128358(CHEMBL3629347)copy SMILEScopy InChI
Affinity DataIC50: 0.160nMAssay Description:Inhibition of human recombinant melanocortin 4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Displacement of [3H]4-DAMP from human recombinant Muscarinic acetylcholine receptor M3 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataIC50: 0.470nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)copy SMILEScopy InChI
Affinity DataIC50: 0.520nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)copy SMILEScopy InChI
Affinity DataIC50: 0.680nMAssay Description:Displacement of [3H]U 69593 from rat recombinant kappa opioid receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)copy SMILEScopy InChI
Affinity DataIC50: 0.810nMAssay Description:Displacement of [3H]methyl-spiperone from human recombinant D2S receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMedDrugBank
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50176062(3-(5H-dibenzo[a,d][7]annulen-5-yl)-N-methylpropan-...)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Displacement of [3H]nisoxetine from human recombinant norepinephrine transporter expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMedDrugBank
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM28582(1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Displacement of [125I](+/-)DOI from human recombinant 5-HT2B receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetSubstance-K receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233962(CHEMBL4068783)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]NKA from human recombinant tachykinin NK2 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50005534(1-(1-(benzo[b]thiophen-2-yl)cyclohexyl)piperidine ...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]BTCP from human recombinant dopamine transporter expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]pirenzepine from human recombinant Muscarinic acetylcholine receptor M1 expressed in CHO cells after 60 mins by scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT5a receptor in HEK293 cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50316543(CHEMBL1094197 | N,N'-(Propane-1,3-diyl)bis(6,7-dih...)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of recombinant dynamin 2 expressed in Sf9 cells by malachite green GTPase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5903PubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50316542(CHEMBL1098764 | N,N'-(Propane-1,3-diyl)bis(7,8-dih...)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant dynamin 2 expressed in Sf9 cells by malachite green GTPase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5903PubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50316539(CHEMBL1094850 | N,N'-(Ethane-1,2-diyl)bis(7,8-dihy...)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Inhibition of recombinant dynamin 2 expressed in Sf9 cells by malachite green GTPase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5903PubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM181119(US9138393, Cimetidine | US9144538, Cimetidine)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Displacement of [125I]APT from human recombinant histamine H2 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233983(CHEMBL4073116)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of phosphatidyl serine liposome-stimulated dynamin 2 GTPase activity (unknown origin) assessed as reduction orthophosphate release using G...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233972(CHEMBL4098509)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of phosphatidyl serine liposome-stimulated dynamin 2 GTPase activity (unknown origin) assessed as reduction orthophosphate release using G...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetDynamin-1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50177941(2-cyano-N-{3-[2-cyano-3-(3,4,5-trihydroxyphenyl)ac...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3Z41PubMed
TargetDynamin-1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM5149((2E)-2-cyano-N-{3-[(2E)-2-cyano-3-(3,4-dihydroxyph...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3Z41PubMed
TargetDynamin-1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50177923(2-cyano-N-{3-[2-cyano-3-(3,4,5-trihydroxyphenyl)ac...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3Z41PubMed
TargetDynamin-1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50177937(2-cyano-N-{3-[2-cyano-3-(3,4,5-trihydroxyphenyl)ac...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3Z41PubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233969(CHEMBL4083788)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of phosphatidyl serine liposome-stimulated dynamin 2 GTPase activity (unknown origin) assessed as reduction orthophosphate release using G...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233975(CHEMBL4064353)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of phosphatidyl serine liposome-stimulated dynamin 2 GTPase activity (unknown origin) assessed as reduction orthophosphate release using G...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50423883(CHEMBL2312430)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of dyn2 in human U2OS cells assessed as clathrin-mediated endocytosis of Tfn after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5GZ3PubMed
TargetDynamin-1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM5152((2E)-2-cyano-N-{4-[(2E)-2-cyano-3-(3,4,5-trihydrox...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3Z41PubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50423885(CHEMBL2312431)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of dyn2 in human U2OS cells assessed as clathrin-mediated endocytosis of Tfn after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5GZ3PubMed
TargetDynamin-1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50147563(CHEMBL109458 | Trimethyl-octadecyl-ammonium; bromi...)copy SMILEScopy InChI
Affinity DataIC50: 3.15E+3nMAssay Description:Concentration required against dynamin-1 GTPase activity of sheep brain.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M07CTPubMed
TargetDynamin-1(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM5151((2E)-2-cyano-N-{4-[(2E)-2-cyano-3-(3,4-dihydroxyph...)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3Z41PubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50423886(CHEMBL2312428)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of dyn2 in human U2OS cells assessed as clathrin-mediated endocytosis of Tfn after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5GZ3PubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50423888(CHEMBL2312414)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of dyn2 in human U2OS cells assessed as clathrin-mediated endocytosis of Tfn after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5GZ3PubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233996(CHEMBL4073407)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of dynamin 2 in human U2OS cells assessed as reduction in clathrin-mediated endocytosis by measuring transferrin-A594 uptake preincubated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
TargetDynamin-2(Homo sapiens (Human))
The University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50233981(CHEMBL4060114)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of phosphatidyl serine liposome-stimulated dynamin 2 GTPase activity (unknown origin) assessed as reduction orthophosphate release using G...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0B6TPubMed
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