Compile Data Set for Download or QSAR
Found 285 with Last Name = 'stephani' and Initial = 'r'
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329839(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329851(3-(3-carboxybenzyl)-1-((6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 0.690nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249533(CHEMBL4078537)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249565(CHEMBL4075238)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at ETB receptor (unknown origin) expressed in HEK293T cells measured after 30 mins by CCF4-AM dye based GeneBlazer FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249532(CHEMBL4061110)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329843(6-Butoxy-3-(3-carboxybenzyl)-1-[(6-ethylbenzo[d][1...)copy SMILEScopy InChI
Affinity DataIC50: 1.44nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329843(6-Butoxy-3-(3-carboxybenzyl)-1-[(6-ethylbenzo[d][1...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329839(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329839(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249531(CHEMBL4081426)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329844(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329838(3-(3-Carboxybenzyl)-6-ethoxy-1-[(6-ethylbenzo[d][1...)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329838(3-(3-Carboxybenzyl)-6-ethoxy-1-[(6-ethylbenzo[d][1...)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249530(CHEMBL4088349)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249564(CHEMBL4095638)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329848(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 7.40nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329845(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329844(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329840(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249529(CHEMBL4067475)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329842(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329842(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 24.4nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)copy SMILEScopy InChI
Affinity DataIC50: 24.8nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50180302(8-(6-iodo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isop...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087810(CHEMBL3426784 | US10428068, Compound 52 | US108440...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of Cy3B-GM from recombinant Hsp90alpha (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249521(CHEMBL4096346)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329837(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329841(6-(Allyloxy)-3-(3-carboxybenzyl)-1-[(6-ethylbenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329841(6-(Allyloxy)-3-(3-carboxybenzyl)-1-[(6-ethylbenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 38.1nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329837(3-(3-Carboxybenzyl)-1-[(6-ethylbenzo[d][1,3]dioxol...)copy SMILEScopy InChI
Affinity DataIC50: 38.9nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50180302(8-(6-iodo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isop...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Displacement of Cy3B-GM from recombinant Hsp90beta (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50180302(8-(6-iodo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isop...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Displacement of Cy3B-GM from recombinant Hsp90alpha (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249563(CHEMBL4100579)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249537(CHEMBL4071505)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087811(CHEMBL3426785)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of Cy3B-GM from recombinant Hsp90alpha (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087810(CHEMBL3426784 | US10428068, Compound 52 | US108440...)copy SMILEScopy InChI
Affinity DataIC50: 101nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329846(3-(3-Carboxybenzyl)-6-(cyclopropylmethoxy)-1-[(6-e...)copy SMILEScopy InChI
Affinity DataIC50: 116nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50165316(8-(2,4-Dichloro-phenylsulfanyl)-9-pent-4-ynyl-9H-p...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329846(3-(3-Carboxybenzyl)-6-(cyclopropylmethoxy)-1-[(6-e...)copy SMILEScopy InChI
Affinity DataIC50: 121nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50165315(9-Pent-4-ynyl-8-(2,4,5-trichloro-phenylsulfanyl)-9...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50180302(8-(6-iodo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isop...)copy SMILEScopy InChI
Affinity DataIC50: 205nMAssay Description:Displacement of PU-FITC3 from recombinant TRAP-1 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087721(CHEMBL3426781)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087447(CHEMBL3426734)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50165268(8-(3,5-Dichloro-phenylsulfanyl)-9-pent-4-ynyl-9H-p...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087811(CHEMBL3426785)copy SMILEScopy InChI
Affinity DataIC50: 265nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50249534(CHEMBL4068786)copy SMILEScopy InChI
Affinity DataIC50: 279nMAssay Description:Antagonist activity at ETA receptor (unknown origin) expressed in membranes by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S21PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
St. John's University

Curated by ChEMBL
LigandPNGBDBM50329849(3-(3-Carboxybenzyl)-6-(carboxymethoxy)-1-[(6-ethyl...)copy SMILEScopy InChI
Affinity DataIC50: 285nMAssay Description:Displacement of [125I]ET1 from ETA receptor expressed in african green monkey CCL-81 cells monolayerMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XPPPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087454(CHEMBL3426741)copy SMILEScopy InChI
Affinity DataIC50: 287nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087448(CHEMBL3426735)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))
Sloan-Kettering

Curated by ChEMBL
LigandPNGBDBM50087575(CHEMBL3426763)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
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