Compile Data Set for Download or QSAR
Found 196 with Last Name = 'einav' and Initial = 's'
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  541nMAssay Description:Binding affinity to biotinylated AAK1 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  1.75E+3nMAssay Description:Binding affinity to biotinylated GAK (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity to biotinylated BMP2K (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetSerine/threonine-protein kinase 16(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  1.19E+4nMAssay Description:Binding affinity to biotinylated STK16 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502299(CHEMBL4544854)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM311155((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-cyanop...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM321107((S)-ethyl (8-((2-amino-2,4-dimethylpentyl)oxy)-6H-...)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562897(CHEMBL4740761)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562898(CHEMBL4778276)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM335593(3-((5-((4-aminopiperidin-1-yl)methyl)pyrrolo[2,1-f...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562894(CHEMBL4762694)copy SMILES
Affinity DataIC50: 3.80nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM279457((R)-1-(5-(7H-pyrrolo[2, 3-d]pyrimidin-4-yl)-1H-ben...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502295(CHEMBL4439128)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502283(CHEMBL4541962)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502285(CHEMBL4543869)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of thrombin-recognition site-fused GST-tagged human AAK1 expressed in bacterial expression system using 5-FAM-Aha-KEEQSQITSQVTGQIGWR-NH2 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562893(CHEMBL4764705)copy SMILES
Affinity DataIC50: 7.70nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562895(CHEMBL4794323)copy SMILES
Affinity DataIC50: 8.80nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502308(CHEMBL4442812)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562914(CHEMBL4745919)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562913(CHEMBL4745028)copy SMILES
Affinity DataIC50: 13nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562905(CHEMBL4800032)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562896(CHEMBL4779229)copy SMILES
Affinity DataIC50: 17nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502304(CHEMBL4483684)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538885(CHEMBL4646895)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50445242(CHEMBL3102941)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538901(CHEMBL4642467)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562907(CHEMBL4752286)copy SMILES
Affinity DataIC50: 35nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562908(CHEMBL4784439)copy SMILES
Affinity DataIC50: 37nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562906(CHEMBL4755134)copy SMILES
Affinity DataIC50: 39nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50288800(CHEMBL4172550)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538879(CHEMBL4645917)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50524284(CHEMBL4443342)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of NanoBRET tracer 5 binding to NL-fused GAK (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50086268(CHEMBL3425867)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562911(CHEMBL4790097)copy SMILES
Affinity DataIC50: 62nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562904(CHEMBL4760106)copy SMILES
Affinity DataIC50: 69nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538876(CHEMBL4642620)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502305(CHEMBL4443908)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538890(CHEMBL4636314)copy SMILEScopy InChI
Affinity DataIC50: 73nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562901(CHEMBL4782363)copy SMILES
Affinity DataIC50: 74nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562915(CHEMBL4756485)copy SMILES
Affinity DataIC50: 78nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562910(CHEMBL4753946)copy SMILES
Affinity DataIC50: 78nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538887(CHEMBL4643096)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50562909(CHEMBL4799769)copy SMILES
Affinity DataIC50: 85nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538900(CHEMBL4641825)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538888(CHEMBL4632903)copy SMILEScopy InChI
Affinity DataIC50: 101nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50045333(CHEBI:90705 | SB-203580)copy SMILES
Affinity DataIC50: 105nMAssay Description:Inhibition of GAK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13D4PubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50502289(CHEMBL4444527)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Displacement of tracer 222 from GST-tagged recombinant human AAK1 catalytic domain (1 to 510 amino acids) expressed in insect cells shaken for 30 sec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50538897(CHEMBL4639991)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
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